SCHEMBL13575002

SCHEMBL13575002

O=C(NC1c2cccc(-c3nc4ccc(F)cc4[nH]3)c2-n2cccc21)C1CC=Nc2[nH]ccc21

nearest known ligand 0.33

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
AMY1A P0DUB6 4/20 0.33
HCRTR1 O43613 1/20 0.32
APAF1 O14727 1/20 0.31
IDO1 P14902 1/20 0.31
BACE1 P56817 2/20 0.31
BACE2 Q9Y5Z0 2/20 0.31
HSP90AB1 P08238 1/20 0.31
F7 P08709 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2158416 0.77 HSP90AB1 (0.56) AMY1AHCRTR1IDO1HSP90AB1
SCHEMBL2159654 0.75 AMY1A (0.43) AMY1AIDO1F7
SCHEMBL13575003 0.75 HSP90AB1 (0.42) HSP90AB1
SCHEMBL14343838 0.75 HSP90AB1 (0.42) AMY1AIDO1BACE1BACE2HSP90AB1
SCHEMBL2747190 0.74 AMY1A (0.43) AMY1AIDO1BACE1BACE2F7
SCHEMBL1550931 0.72 AMY1A (0.47) AMY1AIDO1BACE1BACE2F7
Acetic Acid SCHEMBL2159650 0.72 AMY1A (0.44) AMY1AIDO1F7
SCHEMBL12430611 0.71 HSP90AB1 (0.61) HSP90AB1
SCHEMBL14406022 0.69 HSP90AB1 (0.58) HSP90AB1
SCHEMBL2158386 0.65 HSP90AB1 (0.71) HSP90AB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009153516-A1 NOVEL DERIVATIVES OF PYRROLOINDOLE INHIBITORS OF HSP90, COMPOSITIONS CONTAINING SAME, AND USE THEREOF SANOFI-AVENTIS (FR) 2009-12-23 WO disclosed