SCHEMBL13575003

SCHEMBL13575003

O=C(NC1c2cccc(-c3nc4ccncc4[nH]3)c2-n2cccc21)C1CC(Cl)=Nc2[nH]ccc21

nearest known ligand 0.42

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
HSP90AB1 P08238 4/20 0.42
PDE5A O76074 2/20 0.31
HPSE Q9Y251 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2158650 0.78 HSP90AB1 (0.57) HSP90AB1PDE5AHPSE
SCHEMBL2158386 0.77 HSP90AB1 (0.71) HSP90AB1PDE5AHPSE
SCHEMBL14343938 0.76 HSP90AB1 (0.47) HSP90AB1PDE5AHPSE
SCHEMBL14406022 0.75 HSP90AB1 (0.58) HSP90AB1PDE5AHPSE
SCHEMBL13575002 0.75 AMY1A (0.33) HSP90AB1
SCHEMBL14344002 0.75 HSP90AB1 (0.54) HSP90AB1PDE5AHPSE
SCHEMBL1551437 0.71 HSP90AB1 (0.48) HSP90AB1PDE5AHPSE
SCHEMBL12430611 0.70 HSP90AB1 (0.61) HSP90AB1PDE5AHPSE
SCHEMBL1551252 0.70 PDE5A (0.45) HSP90AB1PDE5AHPSE
SCHEMBL2158416 0.66 HSP90AB1 (0.56) HSP90AB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009153516-A1 NOVEL DERIVATIVES OF PYRROLOINDOLE INHIBITORS OF HSP90, COMPOSITIONS CONTAINING SAME, AND USE THEREOF SANOFI-AVENTIS (FR) 2009-12-23 WO disclosed