SCHEMBL13577014

SCHEMBL13577014

CC(Oc1ccc(F)c(N)c1)c1c(Cl)cccc1Cl

nearest known ligand 0.48

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
MET P08581 15/20 0.48
KDR P35968 6/20 0.48
SRC P12931 3/20 0.48
FGFR2 P21802 2/20 0.48
AXL P30530 2/20 0.48
FLT3 P36888 2/20 0.48
MST1R Q04912 2/20 0.48
KIT P10721 1/20 0.48
INPPL1 O15357 4/20 0.44
AURKA O14965 1/20 0.43
ABL1 P00519 1/20 0.43
LCK P06239 1/20 0.43
FYN P06241 1/20 0.43
YES1 P07947 1/20 0.43
EPHA2 P29317 1/20 0.43
LTK P29376 1/20 0.43
PTK6 Q13882 1/20 0.43
JAK2 O60674 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13577142 0.86 MET (0.42) METKDRSRCFGFR2AXL
SCHEMBL3102747 0.86 NR4A1 (0.41) METKDRSRCFGFR2AXL
SCHEMBL13577013 0.86 MET (0.40) METKDRSRCFGFR2AXL
SCHEMBL13577016 0.84 IGLV6-57 (0.40) METKDRSRCFGFR2AXL
SCHEMBL13577158 0.82 MET (0.45) METKDRSRCFGFR2AXL
SCHEMBL13577019 0.81 DHFR (0.46) METKDRSRCFGFR2AXL
SCHEMBL3101898 0.80 MET (0.58) METKDRSRCFGFR2AXL
SCHEMBL4301190 0.79 GNRHR (0.46) METKDRSRCFGFR2AXL
SCHEMBL13577182 0.78 CYP3A4 (0.47) METKDRSRCFGFR2AXL
SCHEMBL3097665 0.78 MET (0.47) METINPPL1JAK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9040693-B2 Fused heterocyclic derivative, medicinal composition containing the same, and medicinal use thereof KISSEI PHARMACEUTICAL CO., LTD. (JP) 2015-05-26 US disclosed
US-9040693-B2 Fused heterocyclic derivative, medicinal composition containing the same, and medicinal use thereof KISSEI PHARMACEUTICAL CO., LTD. (JP) 2015-05-26 US disclosed
US-20090325900-A1 FUSED HETEROCYCLIC DERIVATIVE, MEDICINAL COMPOSITION CONTAINING THE SAME, AND MEDICINAL USE THEREOF KISSEI PHARMACEUTICAL CO., LTD. (JP) 2009-12-31 US disclosed
US-20090325900-A1 FUSED HETEROCYCLIC DERIVATIVE, MEDICINAL COMPOSITION CONTAINING THE SAME, AND MEDICINAL USE THEREOF KISSEI PHARMACEUTICAL CO., LTD. (JP) 2009-12-31 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090325900-A1 FUSED HETEROCYCLIC DERIVATIVE, MEDICINAL COMPOSITION CONTAINING THE SAME, AND MEDICINAL USE THEREOF SHBG, CYP19A1, NR5A1 MET 202/4885KDR 1862/4885SRC 1086/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.