SCHEMBL1358320

SCHEMBL1358320

CC(C)(C)c1cc(-c2ccc[nH]c2=O)cc2c(C(=O)N3CCC(C(N)=O)CC3)coc12

nearest known ligand 0.39

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.39
SMN1; SMN2 Q16637 3/20 0.37
PKM P14618 1/20 0.37
NPC1 O15118 4/20 0.35
RAB9A P51151 3/20 0.35
KMT2A Q03164 1/20 0.35
TDP1 Q9NUW8 2/20 0.35
GAA P10253 1/20 0.35
BRD9 Q9H8M2 1/20 0.34
POLB P06746 1/20 0.33
HSD17B10 Q99714 1/20 0.33
CYP3A4 P08684 1/20 0.33
PARP1 P09874 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3144828 0.95 PDK2 (0.36) ALDH1A1SMN1; SMN2PKMNPC1RAB9A
SCHEMBL1360205 0.91 KDM1A (0.38) CYP3A4
SCHEMBL1357846 0.91 HSP90AA1 (0.40) GAACYP3A4
SCHEMBL1359379 0.90 RAB9A (0.39) ALDH1A1NPC1RAB9ATDP1GAA
SCHEMBL1359385 0.89 MAPT (0.36) ALDH1A1SMN1; SMN2KMT2AGAAPOLB
SCHEMBL1359911 0.89 MAPT (0.34) ALDH1A1SMN1; SMN2KMT2AGAAPOLB
SCHEMBL1358259 0.88 KDM1A (0.37) CYP3A4PARP1
SCHEMBL1359529 0.88 MAPT (0.37) ALDH1A1SMN1; SMN2NPC1RAB9AKMT2A
SCHEMBL1359618 0.87 CHEK1 (0.42) GAACYP3A4
SCHEMBL1358783 0.87 HSP90AA1 (0.39) ALDH1A1SMN1; SMN2GAABRD9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8067442-B2 Heterocyclic antiviral compounds ROCHE PALO ALTO LLC (US) 2011-11-29 US claimed
EP-2334662-A1 PYRINE OR PYRAZINE DERIVATIVES FOR TREATING HCV F. Hoffmann-La Roche AG (CH) 2011-06-22 EP claimed
US-20100081658-A1 HETEROCYCLIC ANTIVIRAL COMPOUNDS ROCHE PALO ALTO LLC 2010-04-01 US claimed
WO-2010034671-A1 PYRINE OR PYRAZINE DERIVATIVES FOR TREATING HCV F. HOFFMANN-LA ROCHE AG (CH) 2010-04-01 WO claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100081658-A1 HETEROCYCLIC ANTIVIRAL COMPOUNDS EIF2AK2, POLR2A, HCCS ALDH1A1 1038/4885SMN1; SMN2 3473/4885PKM 3533/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.