SCHEMBL1359862

SCHEMBL1359862

Cn1cc(C#N)c2cc(-c3ccc[nH]c3=O)cc(C(C)(C)C)c21

nearest known ligand 0.39

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
MCL1 Q07820 4/20 0.39
CYP3A4 P08684 3/20 0.36
KDM4E B2RXH2 6/20 0.36
ALDH1A1 P00352 6/20 0.36
GAA P10253 4/20 0.36
GLA P06280 1/20 0.36
BRD4 O60885 3/20 0.35
IMPDH2 P12268 1/20 0.34
HPGD P15428 2/20 0.32
PRMT5 O14744 1/20 0.32
WDR77 Q9BQA1 1/20 0.32
CYP1A2 P05177 1/20 0.31
BRD9 Q9H8M2 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1359429 0.80 CYP3A4 (0.36) CYP3A4KDM4EBRD4
SCHEMBL1971791 0.78 IMPDH2 (0.47) MCL1KDM4EALDH1A1BRD4IMPDH2
SCHEMBL1358987 0.75 CYP3A4 (0.40) CYP3A4KDM4EALDH1A1GAABRD4
SCHEMBL1359884 0.69 CYP3A4 (0.35) MCL1CYP3A4
SCHEMBL12138690 0.69 CHEK1 (0.37) CYP3A4BRD4
SCHEMBL1357997 0.69 CYP3A4 (0.40) MCL1CYP3A4
SCHEMBL1543883 0.68 CYP3A4 (0.61) MCL1CYP3A4KDM4EALDH1A1GAA
SCHEMBL1360035 0.68 BRD4 (0.40) CYP3A4BRD4
SCHEMBL1543881 0.68 CYP3A4 (0.61) MCL1CYP3A4KDM4EALDH1A1GAA
SCHEMBL1358251 0.65 CYP3A4 (0.38) CYP3A4KDM4EALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8067442-B2 Heterocyclic antiviral compounds ROCHE PALO ALTO LLC (US) 2011-11-29 US claimed
US-20100081658-A1 HETEROCYCLIC ANTIVIRAL COMPOUNDS ROCHE PALO ALTO LLC 2010-04-01 US claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100081658-A1 HETEROCYCLIC ANTIVIRAL COMPOUNDS EIF2AK2, POLR2A, HCCS MCL1 2162/4885CYP3A4 713/4885KDM4E 2198/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.