SCHEMBL1360027

SCHEMBL1360027

CC(C)S(=O)(=O)NC[C@H]1CCN(C(=O)c2coc3c(C(C)(C)C)cc(-c4ccc[nH]c4=O)cc23)C1

nearest known ligand 0.33

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
NPY5R Q15761 4/20 0.33
CYP3A4 P08684 3/20 0.33
F10 P00742 1/20 0.33
BRD4 O60885 1/20 0.32
RORC P51449 1/20 0.32
ALDH1A1 P00352 1/20 0.30
KCNH2 Q12809 1/20 0.30
SMYD3 Q9H7B4 1/20 0.30
USP9X Q93008 1/20 0.30
TGFBR1 P36897 1/20 0.30
TLR9 Q9NR96 1/20 0.30
TLR8 Q9NR97 1/20 0.30
TLR7 Q9NYK1 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1359499 0.93 CYP3A4 (0.37) CYP3A4F10BRD4RORCALDH1A1
SCHEMBL1358011 0.93 CYP3A4 (0.37) CYP3A4F10BRD4RORCALDH1A1
SCHEMBL1360041 0.92 CYP3A4 (0.34) CYP3A4F10BRD4RORCALDH1A1
SCHEMBL1360367 0.92 CYP3A4 (0.34) CYP3A4F10BRD4RORCALDH1A1
SCHEMBL1359241 0.89 ALDH1A1 (0.36) CYP3A4ALDH1A1
SCHEMBL1358409 0.89 ALDH1A1 (0.36) CYP3A4ALDH1A1
SCHEMBL1360029 0.89 ALDH1A1 (0.36) CYP3A4ALDH1A1
SCHEMBL1359531 0.88 KCNH2 (0.33) CYP3A4KCNH2
SCHEMBL1360760 0.87 HTR2C (0.36) CYP3A4RORC
SCHEMBL1972033 0.87 CYP3A4 (0.39) CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8067442-B2 Heterocyclic antiviral compounds ROCHE PALO ALTO LLC (US) 2011-11-29 US claimed