SCHEMBL1360041

SCHEMBL1360041

CCS(=O)(=O)NC[C@H]1CCN(C(=O)c2coc3c(C(C)(C)C)cc(-c4ccc[nH]c4=O)cc23)C1

nearest known ligand 0.34

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 3/20 0.34
BRD4 O60885 1/20 0.33
RORC P51449 1/20 0.33
F10 P00742 1/20 0.32
ALDH1A1 P00352 2/20 0.31
TGFBR1 P36897 1/20 0.30
TDP1 Q9NUW8 1/20 0.30
HTR2C P28335 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1358011 0.93 CYP3A4 (0.37) CYP3A4BRD4RORCF10ALDH1A1
SCHEMBL1359499 0.93 CYP3A4 (0.37) CYP3A4BRD4RORCF10ALDH1A1
SCHEMBL1360367 0.93 CYP3A4 (0.34) CYP3A4BRD4RORCF10ALDH1A1
SCHEMBL1360027 0.92 NPY5R (0.33) CYP3A4BRD4RORCF10ALDH1A1
SCHEMBL1358409 0.89 ALDH1A1 (0.36) CYP3A4ALDH1A1TDP1
SCHEMBL1359241 0.89 ALDH1A1 (0.36) CYP3A4ALDH1A1TDP1
SCHEMBL1360029 0.89 ALDH1A1 (0.36) CYP3A4ALDH1A1TDP1
SCHEMBL1359531 0.89 KCNH2 (0.33) CYP3A4HTR2C
SCHEMBL1360760 0.88 HTR2C (0.36) CYP3A4RORCHTR2C
SCHEMBL1972033 0.87 CYP3A4 (0.39) CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8067442-B2 Heterocyclic antiviral compounds ROCHE PALO ALTO LLC (US) 2011-11-29 US claimed