SCHEMBL1360132

SCHEMBL1360132

CC(C)(C)c1cc(-c2ccc[nH]c2=O)cc2c(C(=O)N3CC(O)C3)coc12

nearest known ligand 0.35

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 3/20 0.35
CHEK1 O14757 2/20 0.34
ALOX5AP P20292 1/20 0.32
FEN1 P39748 1/20 0.32
MAP4K4 O95819 1/20 0.32
GAA P10253 1/20 0.32
PDK2 Q15119 2/20 0.31
HSP90AA1 P07900 1/20 0.30
HSP90AB1 P08238 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1359618 0.93 CHEK1 (0.42) CYP3A4CHEK1ALOX5APFEN1GAA
SCHEMBL1357846 0.92 HSP90AA1 (0.40) CYP3A4CHEK1ALOX5APFEN1GAA
SCHEMBL1359797 0.91 CHEK1 (0.38) CYP3A4CHEK1ALOX5APFEN1GAA
SCHEMBL1360377 0.90 CHEK1 (0.34) CYP3A4CHEK1GAAPDK2
SCHEMBL1359911 0.89 MAPT (0.34) CYP3A4GAA
SCHEMBL1359385 0.89 MAPT (0.36) CYP3A4GAA
SCHEMBL1359529 0.88 MAPT (0.37) CYP3A4GAA
SCHEMBL1358783 0.87 HSP90AA1 (0.39) ALOX5APGAAHSP90AA1HSP90AB1
SCHEMBL1359635 0.87 HSP90AA1 (0.38) CYP3A4HSP90AA1HSP90AB1
SCHEMBL1358259 0.87 KDM1A (0.37) CYP3A4CHEK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8067442-B2 Heterocyclic antiviral compounds ROCHE PALO ALTO LLC (US) 2011-11-29 US claimed
EP-2334662-A1 PYRINE OR PYRAZINE DERIVATIVES FOR TREATING HCV F. Hoffmann-La Roche AG (CH) 2011-06-22 EP claimed
US-20100081658-A1 HETEROCYCLIC ANTIVIRAL COMPOUNDS ROCHE PALO ALTO LLC 2010-04-01 US claimed
WO-2010034671-A1 PYRINE OR PYRAZINE DERIVATIVES FOR TREATING HCV F. HOFFMANN-LA ROCHE AG (CH) 2010-04-01 WO claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100081658-A1 HETEROCYCLIC ANTIVIRAL COMPOUNDS EIF2AK2, POLR2A, HCCS CYP3A4 713/4885CHEK1 1363/4885ALOX5AP 3018/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.