SCHEMBL13602811

SCHEMBL13602811

N#Cc1ccc(-n2ccc(O)cc2=O)cc1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 1/20 0.45
CA2 P00918 1/20 0.45
CA3 P07451 1/20 0.45
CA6 P23280 1/20 0.45
CA9 Q16790 1/20 0.45
CA14 Q9ULX7 1/20 0.45
TRPV1 Q8NER1 1/20 0.42
CYP19A1 P11511 1/20 0.42
POLB P06746 1/20 0.41
MMP3 P08254 1/20 0.41
CYP11B2 P19099 3/20 0.39
PKM P14618 1/20 0.39
ELANE P08246 1/20 0.38
ESRRA P11474 1/20 0.38
ALDH1A1 P00352 1/20 0.38
ALOX15 P16050 1/20 0.38
HTT P42858 1/20 0.38
ATM Q13315 1/20 0.38
GPR119 Q8TDV5 1/20 0.37
MAOA P21397 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2333255 0.79 CASP3 (0.39) CA12CA2CA3CA6CA9
SCHEMBL12927339 0.77 F2 (0.47) POLBELANEALDH1A1ALOX15HTT
SCHEMBL17979345 0.77 SCD (0.43) ALDH1A1ALOX15HTTATM
SCHEMBL10059741 0.76 SMN1; SMN2 (0.60) ESRRAALDH1A1ALOX15HTTATM
SCHEMBL85902 0.73 HTR1A (0.46) CYP19A1POLBCYP11B2PKMELANE
SCHEMBL10078773 0.72 CA12 (0.50) CA12CA2CA3CA6CA9
SCHEMBL4379409 0.71 MCHR1 (0.65) MAOB
SCHEMBL1550632 0.71 ENPP2 (0.50) ALDH1A1ALOX15HTTATMGPR119
SCHEMBL17979531 0.71 MCHR1 (0.53)
SCHEMBL5576893 0.67 CA12 (0.50) CA12CA2CA3CA6CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7629363-B2 antiinflammatory agent for treating asthma and chronic pulmonary inflammatory disease PFIZER INC (US) 2009-12-08 US disclosed
US-7629363-B2 antiinflammatory agent for treating asthma and chronic pulmonary inflammatory disease PFIZER INC (US) 2009-12-08 US disclosed
EP-1490064-B1 SUBSTITUTED PYRIDINONES AS MODULATORS OF P38 MAP KINASE PHARMACIA CORP (US) 2009-11-18 EP disclosed