SCHEMBL13613557

SCHEMBL13613557

NC(=O)c1c(N)[nH]c2cc(N(O)O)ccc12

nearest known ligand 0.31

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 1/20 0.31
KDM4E B2RXH2 1/20 0.31
ALDH1A1 P00352 1/20 0.31
MAP2 P11137 1/20 0.31
MITF O75030 1/20 0.31
MAPT P10636 1/20 0.31
MEN1 O00255 1/20 0.30
GAA P10253 1/20 0.30
CACNA1B Q00975 1/20 0.30
APBA1 Q02410 1/20 0.30
KMT2A Q03164 1/20 0.30
AR P10275 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3834396 0.86 AR (0.43) PARP1KDM4EALDH1A1MAP2MAPT
SCHEMBL3217527 0.78 FEN1 (0.44) PARP1KDM4EALDH1A1MAP2MEN1
SCHEMBL3210534 0.78 PDPK1 (0.42) PARP1
SCHEMBL3197903 0.78 CA1 (0.49) PARP1KDM4EALDH1A1MAP2MEN1
SCHEMBL3828991 0.78 MITF (0.51) KDM4EALDH1A1MITFMAPTGAA
SCHEMBL3833775 0.77 KMT2A (0.37) ALDH1A1KMT2A
SCHEMBL349187 0.76 PARP1 (0.49) PARP1KDM4EALDH1A1GAAKMT2A
SCHEMBL14236512 0.75 KDR (0.42) KDM4EALDH1A1MAPTGAA
SCHEMBL15146065 0.74 PIN1 (0.41) PARP1MAP2AR
SCHEMBL3197218 0.74 KIF11 (0.55) ALDH1A1MAPTMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2119703-A1 NOVEL INDOLE DERIVATIVE HAVING INHIBITORY ACTIVITY ON I B KINASE Santen Pharmaceutical Co., Ltd (JP) 2009-11-18 EP disclosed