SCHEMBL13613844

SCHEMBL13613844

C#Cc1cc(C(=O)OC(C)C)cc(-c2ccc(CC(=O)O)c(F)c2)c1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CD274 Q9NZQ7 2/20 0.38
PDCD1 Q15116 1/20 0.38
RXRA P19793 3/20 0.37
RXRB P28702 3/20 0.37
RXRG P48443 2/20 0.37
GLRA3 O75311 1/20 0.37
GLRB P48167 1/20 0.37
CA12 O43570 3/20 0.35
CA1 P00915 3/20 0.35
CA2 P00918 3/20 0.35
CA7 P43166 3/20 0.35
CA9 Q16790 3/20 0.35
CA14 Q9ULX7 3/20 0.35
NR1H4 Q96RI1 1/20 0.34
PTPN11 Q06124 1/20 0.33
BDKRB1 P46663 3/20 0.32
CYP4F2 P78329 1/20 0.32
CYP4A11 Q02928 1/20 0.32
FFAR4 Q5NUL3 2/20 0.31
ROCK2 O75116 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13613952 0.86 GLRA3 (0.34) CD274PDCD1GLRA3GLRBCA12
SCHEMBL4519235 0.85 FFAR1 (0.41) FFAR4
SCHEMBL13613914 0.82 PDCD1 (0.49) CD274PDCD1RXRARXRBRXRG
SCHEMBL13613966 0.81 CD274 (0.36) CD274PDCD1RXRARXRBRXRG
SCHEMBL13606700 0.76 FFAR1 (0.41) FFAR4
SCHEMBL4516332 0.75 FFAR1 (0.49) FFAR4NPC1MAPTHTTRAB9A
SCHEMBL4515497 0.73 CA12 (0.56) CD274PDCD1GLRA3GLRBCA12
SCHEMBL4504892 0.72 FFAR1 (0.33) CA12CA1CA2CA7CA9
SCHEMBL5706347 0.70 FFAR1 (0.32) FFAR4
SCHEMBL13613968 0.69 ROCK2 (0.33) CD274PDCD1CA12CA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7638648-B2 Compounds having selective cytochrome P450RAI-1 or selective cytochrome P450RAI-2 inhibitory activity and methods of obtaining the same ALLERGAN INC. (US) 2009-12-29 US disclosed
US-7468391-B2 Methods for treating retinoid responsive disorders using selective inhibitors of CYP26A and CYP26B ALLERGAN, INC. (US) 2008-12-23 US disclosed
US-20080004455-A1 Compounds having selective cytochrome P450RAI-1 or selective cytochrome P450RAI-2 inhibitory activity and methods of obtaining the same ALLERGAN, INC. (US) 2008-01-03 US disclosed
US-7226951-B2 Compounds having selective cytochrome P450RAI-1 or selective cytochrome P450RAI-2 inhibitory activity and methods of obtaining the same ALLERGAN, INC. (US) 2007-06-05 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080004455-A1 Compounds having selective cytochrome P450RAI-1 or selective cytochrome P450RAI-2 inhibitory activity and methods of obtaining the same CYP1A2, CYP2A7, CYP3A7 CD274 4649/4885PDCD1 4633/4885RXRA 351/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.