SCHEMBL1361412

SCHEMBL1361412

CCCC(=O)OCc1cc(C#N)ccc1CCCC(O)(c1ccc(F)cc1)N(C)C

nearest known ligand 0.34

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CXCR2 P25025 10/20 0.34
CYP2C9 P11712 1/20 0.34
NSD2 O96028 1/20 0.32
TBXA2R P21731 1/20 0.31
NR3C1 P04150 1/20 0.31
PGR P06401 1/20 0.31
NR3C2 P08235 1/20 0.31
SLC6A4 P31645 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5718374 0.95 CXCR2 (0.34) CXCR2CYP2C9NSD2NR3C1PGR
SCHEMBL1360673 0.83 KMT2A (0.32) CXCR2CYP2C9
SCHEMBL1561187 0.82 NR3C1 (0.34) CXCR2CYP2C9NSD2NR3C1PGR
SCHEMBL5718466 0.82 NR3C1 (0.34) CXCR2CYP2C9NSD2NR3C1PGR
SCHEMBL2866617 0.82 NR3C1 (0.34) CXCR2CYP2C9NSD2NR3C1PGR
Bromide SCHEMBL4625572 0.81 CXCR2 (0.34) CXCR2CYP2C9NSD2NR3C1PGR
SCHEMBL1363413 0.78 SLC6A4 (0.36) CYP2C9SLC6A4
SCHEMBL1363412 0.78 SLC6A4 (0.36) CYP2C9SLC6A4
SCHEMBL1361410 0.78 NSD2 (0.31) CXCR2CYP2C9NSD2TBXA2RSLC6A4
Benzoic Acid SCHEMBL1360672 0.73 MRGPRX4 (0.33)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8067640-B2 Method for the separation of intermediates which may be used for the preparation of escitalopram H. LUNDBECK A/S (DK) 2011-11-29 US disclosed
US-20110065937-A1 METHOD FOR THE SEPARATION OF INTERMEDIATES WHICH MAY BE USED FOR THE PREPARATION OF ESCITALOPRAM H. LUNDBECK A/S (DK) 2011-03-17 US disclosed
US-20070129561-A1 Method for the separation of intermediates which may be used for the preparation of escitalopram H. LUNDBECK A/S (DK) 2007-06-07 US disclosed
EP-1716108-A1 METHOD FOR THE SEPARATION OF INTERMEDIATES WHICH MAY BE USED FOR THE PREPARATION OF ESCITALOPRAM H. Lundbeck A/S (DK) 2006-11-02 EP disclosed
WO-2005077891-A1 METHOD FOR THE SEPARATION OF INTERMEDIATES WHICH MAY BE USED FOR THE PREPARATION OF ESCITALOPRAM H. LUNDBECK A/S (DK) 2005-08-25 WO disclosed
EP-1534654-A1 METHOD FOR THE SEPARATION OF INTERMEDIATES WHICH MAY BE USED FOR THE PREPARATION OF ESCITALOPRAM H. LUNDBECK A/S (DK) 2005-06-01 EP disclosed
WO-2004014821-A1 METHOD FOR THE SEPARATION OF INTERMEDIATES WHICH MAY BE USED FOR THE PREPARATION OF ESCITALOPRAM H. LUNDBECK A/S (DK) 2004-02-19 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110065937-A1 METHOD FOR THE SEPARATION OF INTERMEDIATES WHICH MAY BE USED FOR THE PREPARATION OF ESCITALOPRAM MAOB, HSD17B14, MAOA CXCR2 3901/4885CYP2C9 29/4885NSD2 1001/4885
US-20070129561-A1 Method for the separation of intermediates which may be used for the preparation of escitalopram MAOB, HSD17B14, MAOA CXCR2 3901/4885CYP2C9 29/4885NSD2 1001/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.