SCHEMBL13617326

SCHEMBL13617326

CC(C)(C)c1c(O)cc([N+](=O)[O-])cc1[N+](=O)[O-]

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GPR35 Q9HC97 8/20 0.59
ALDH1A1 P00352 5/20 0.59
KMT2A Q03164 4/20 0.59
MEN1 O00255 3/20 0.59
HPGD P15428 2/20 0.59
MAPK1 P28482 2/20 0.59
MAPT P10636 2/20 0.59
KDM4E B2RXH2 1/20 0.59
TTR P02766 1/20 0.59
CYP1A2 P05177 1/20 0.59
CYP2C9 P11712 1/20 0.59
ALOX15 P16050 1/20 0.59
ALOX12 P18054 1/20 0.59
RECQL P46063 1/20 0.59
PMP22 Q01453 1/20 0.59
HIF1A Q16665 1/20 0.59
HSD17B10 Q99714 1/20 0.59
TDP1 Q9NUW8 1/20 0.59
HTT P42858 3/20 0.53
SMN1; SMN2 Q16637 2/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4926322 0.87 KMT2A (0.52) GPR35ALDH1A1KMT2AMEN1HPGD
SCHEMBL18688897 0.82 SMN1; SMN2 (0.68) GPR35ALDH1A1KMT2AMEN1HPGD
SCHEMBL13616905 0.78 CA1 (0.49) GPR35ALDH1A1KMT2AMEN1HPGD
SCHEMBL3077511 0.77 ALDH1A1 (0.62) GPR35ALDH1A1KMT2AMEN1HPGD
SCHEMBL3132904 0.76 GPR35 (0.66) GPR35ALDH1A1KMT2AMEN1HPGD
SCHEMBL29577133 0.76 GPR35 (0.66) GPR35ALDH1A1KMT2AMEN1HPGD
Dinoterb SCHEMBL8535102 0.75 KMT2A (0.79) GPR35ALDH1A1KMT2AMEN1HPGD
Dinoterb SCHEMBL53794 0.75 KMT2A (0.79) GPR35ALDH1A1KMT2AMEN1HPGD
Dinoterb SCHEMBL29487271 0.75 KMT2A (0.79) GPR35ALDH1A1KMT2AMEN1HPGD
3,5-Dinitrocatechol (Or-486) SCHEMBL1283419 0.75 GPR35 (1.00) GPR35ALDH1A1KMT2AMEN1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8455497-B2 Inhibitors of aspartyl protease VERTEX PHARMACEUTICALS INCORPORATED (US) 2013-06-04 US disclosed
US-20090274650-A1 INHIBITORS OF ASPARTYL PROTEASE VERTEX PHARMACEUTICALS INCORPORATED 2009-11-05 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090274650-A1 INHIBITORS OF ASPARTYL PROTEASE SPINT2, DNPEP, PRSS1 GPR35 4694/4885ALDH1A1 1604/4885KMT2A 864/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.