SCHEMBL13617435

SCHEMBL13617435

COC(=O)[C@H](Cc1cn(CCc2ccccn2)cn1)NC(=O)OC(C)(C)C

nearest known ligand 0.46

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
HDAC6 Q9UBN7 4/20 0.46
HDAC1 Q13547 2/20 0.46
NLRP3 Q96P20 1/20 0.42
KLK5 Q9Y337 1/20 0.41
SIRT2 Q8IXJ6 9/20 0.39
CPB2 Q96IY4 2/20 0.38
CPB1 P15086 1/20 0.38
TACR1 P25103 1/20 0.38
AKT1 P31749 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3845713 0.91 CPB2 (0.45) CPB2CPB1AKT1
SCHEMBL8345705 0.89 KLK5 (0.49) KLK5SIRT2CPB2CPB1AKT1
SCHEMBL16464699 0.85 HDAC6 (0.60) HDAC6HDAC1NLRP3KLK5TACR1
SCHEMBL16464697 0.85 HDAC6 (0.60) HDAC6HDAC1NLRP3KLK5TACR1
SCHEMBL8347877 0.84 CPB2 (0.54) KLK5SIRT2CPB2CPB1TACR1
SCHEMBL19508750 0.82 KLK5 (0.51) KLK5SIRT2AKT1
SCHEMBL8349511 0.82 CPB2 (0.42) KLK5SIRT2CPB2CPB1TACR1
SCHEMBL6324267 0.81 ACE (0.52) CPB2CPB1AKT1
SCHEMBL8364520 0.79 CPB2 (0.37) KLK5CPB2CPB1TACR1AKT1
SCHEMBL13617417 0.78 CPB2 (0.48) KLK5SIRT2CPB2CPB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1311488-B1 SUBSTITUTED IMIDAZOLES AS TAFIA INHIBITORS PFIZER LTD (GB) 2009-11-04 EP disclosed