SCHEMBL13617547

SCHEMBL13617547

NCCOc1c(F)ccc(F)c1Cl

nearest known ligand 0.41

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
PLAU P00749 2/20 0.41
PARP1 P09874 6/20 0.40
PARP3 Q9Y6F1 6/20 0.40
TAAR1 Q96RJ0 1/20 0.39
KDM4E B2RXH2 1/20 0.39
HTR2C P28335 4/20 0.39
HTR2B P41595 4/20 0.39
HTR2A P28223 3/20 0.39
REN P00797 1/20 0.34
LTA4H P09960 1/20 0.34
PLA2G2A P14555 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL65300 0.82 HTR2A (0.32) HTR2CHTR2BHTR2A
SCHEMBL21601405 0.76 TAAR1 (0.48) PLAUPARP1PARP3TAAR1KDM4E
SCHEMBL24096249 0.76 TAAR1 (0.48) PLAUPARP1PARP3TAAR1KDM4E
SCHEMBL773452 0.74 TSHR (0.47)
Hydrochloric Acid SCHEMBL7484053 0.74 KDM4E (0.52) PARP1TAAR1KDM4EHTR2CHTR2B
SCHEMBL91267 0.72 LMNA (0.43) KDM4E
SCHEMBL661082 0.72 REN (0.40) TAAR1HTR2AREN
SCHEMBL7606607 0.72 REN (0.41) TAAR1REN
SCHEMBL78179 0.71 KDM4E (0.43) KDM4E
SCHEMBL27337036 0.71 HTR2A (0.31) PLAUPARP1PARP3HTR2CHTR2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1888538-B1 (3,4-DIHYDRO-QUINAZOLIN-2-YL)-(2-ARYLOXY-ETHYL)-AMINES HAVING AN ACTIVITY ON THE 5-HT RECEPTOR HOFFMANN LA ROCHE (CH) 2009-11-18 EP disclosed