SCHEMBL65300

SCHEMBL65300

Fc1ccc(F)c(OCCBr)c1Cl

nearest known ligand 0.32

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 3/20 0.32
HTR2C P28335 3/20 0.32
HTR2B P41595 3/20 0.32
EGFR P00533 1/20 0.32
SLC6A2 P23975 4/20 0.30
SLC6A4 P31645 4/20 0.30
SLC6A3 Q01959 4/20 0.30
CYP2D6 P10635 2/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13617547 0.82 PLAU (0.41) HTR2AHTR2CHTR2B
SCHEMBL3119777 0.77 SCN8A (0.36) SLC6A2SLC6A4SLC6A3
SCHEMBL27337036 0.77 HTR2A (0.31) HTR2AHTR2CHTR2B
SCHEMBL661082 0.74 REN (0.40) HTR2A
SCHEMBL27341101 0.71 TDP1 (0.40) HTR2AHTR2CHTR2B
SCHEMBL9142141 0.71
SCHEMBL91267 0.71 LMNA (0.43) CYP2D6
SCHEMBL7606607 0.71 REN (0.41)
SCHEMBL16178976 0.71 SCN8A (0.33)
SCHEMBL78179 0.70 KDM4E (0.43)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8129538-B1 Renin inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2012-03-06 US disclosed
US-8129538-B1 Renin inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2012-03-06 US disclosed
US-8129538-B1 Renin inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2012-03-06 US disclosed