SCHEMBL13618169

SCHEMBL13618169

COc1cc(C)cc(CCCc2cc(O)cc(OC)c2)c1

nearest known ligand 0.68

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 4/20 0.68
CALM1 P0DP23 6/20 0.61
GABRA1 P14867 1/20 0.57
GABRG2 P18507 1/20 0.57
GABRB3 P28472 1/20 0.57
GABRA3 P34903 1/20 0.57
GABRA2 P47869 1/20 0.57
GABRB2 P47870 1/20 0.57
PTPN1 P18031 2/20 0.53
NOS2 P35228 1/20 0.53
AKR1B1 P15121 2/20 0.48
BACE1 P56817 1/20 0.45
CYP3A4 P08684 2/20 0.43
ESR1 P03372 1/20 0.43
CYP19A1 P11511 1/20 0.43
ESR2 Q92731 1/20 0.43
TACR1 P25103 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24076843 0.89 CALM1 (0.64) PTGS2CALM1GABRA1GABRG2GABRB3
SCHEMBL10186605 0.81 PTGS2 (0.70) PTGS2CALM1GABRA1GABRG2GABRB3
SCHEMBL10654346 0.81 PTGS2 (1.00) PTGS2CALM1GABRA1GABRG2GABRB3
SCHEMBL17509775 0.79 PTGS2 (0.97) PTGS2CALM1GABRA1GABRG2GABRB3
SCHEMBL21925060 0.79 PTGS2 (0.97) PTGS2CALM1GABRA1GABRG2GABRB3
SCHEMBL17509787 0.79 PTGS2 (0.97) PTGS2CALM1GABRA1GABRG2GABRB3
SCHEMBL23462775 0.79 PTGS2 (0.97) PTGS2CALM1GABRA1GABRG2GABRB3
SCHEMBL10296730 0.79 PTGS2 (0.50) PTGS2CALM1GABRA1GABRG2GABRB3
SCHEMBL10652400 0.79 PTGS2 (0.97) PTGS2CALM1GABRA1GABRG2GABRB3
SCHEMBL20179619 0.79 CALM1 (0.65) PTGS2CALM1GABRA1GABRG2GABRB3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1833816-B1 SUBSTITUTED PIPERIDINES AS RENIN INHIBITORS NOVARTIS AG (CH) 2009-11-11 EP disclosed