SCHEMBL13618755

SCHEMBL13618755

NC(=O)c1cc(Br)ccc1NC=O

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DGAT1 O75907 1/20 0.47
IRAK4 Q9NWZ3 1/20 0.41
KDM4E B2RXH2 3/20 0.41
GLA P06280 2/20 0.41
ALDH1A1 P00352 2/20 0.41
MAP2K1 Q02750 2/20 0.40
KDM5A P29375 2/20 0.40
MAP2K2 P36507 1/20 0.40
GAA P10253 1/20 0.40
APEX1 P27695 1/20 0.40
PLAU P00749 1/20 0.39
CES2 O00748 1/20 0.39
GALR3 O60755 1/20 0.39
CYP1A2 P05177 1/20 0.39
CYP2C9 P11712 1/20 0.39
HPGD P15428 1/20 0.39
ALOX15 P16050 1/20 0.39
CASP1 P29466 1/20 0.39
CYP2C19 P33261 1/20 0.39
MAPT P10636 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10082578 0.86 DGAT1 (0.51) DGAT1KDM4EGLAALDH1A1MAP2K1
SCHEMBL7806435 0.81 KDM5A (0.45) KDM4EGLAALDH1A1KDM5AGAA
SCHEMBL21666210 0.79 ALDH1A1 (0.64) DGAT1IRAK4KDM4EGLAALDH1A1
SCHEMBL21075953 0.78 ALDH1A1 (0.43) KDM4EGLAALDH1A1KDM5AGAA
SCHEMBL22101252 0.78 ALDH1A1 (0.43) KDM4EALDH1A1KDM5AGAAAPEX1
SCHEMBL17540395 0.77 DGAT1 (0.41) DGAT1KDM4EALDH1A1MAP2K1KDM5A
SCHEMBL27959043 0.76 DGAT1 (0.47) DGAT1IRAK4KDM4EGLAALDH1A1
SCHEMBL26170005 0.76 ALDH1A1 (0.69) DGAT1IRAK4KDM4EGLAALDH1A1
SCHEMBL13167870 0.74 AAK1 (0.45) KDM4EGLAALDH1A1KDM5AMAPT
SCHEMBL2612359 0.74 KDM4E (0.58) KDM4EALDH1A1GAAHPGDCASP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009143049-A1 BICYCLIC HETEROCYCLE DERIVATIVES AND USE THEREOF AS GPR119 MODULATORS SCHERING CORPORATION (US) 2009-11-26 WO disclosed