SCHEMBL22101252

SCHEMBL22101252

C=C(C)c1cc(Br)ccc1NC=O

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.43
OR51E2 Q9H255 1/20 0.37
STAT3 P40763 5/20 0.36
KDM5A P29375 1/20 0.36
APEX1 P27695 1/20 0.36
POLB P06746 3/20 0.35
MEN1 O00255 3/20 0.35
KMT2A Q03164 3/20 0.35
MAPT P10636 4/20 0.35
GAA P10253 3/20 0.35
HTT P42858 2/20 0.35
KDM4E B2RXH2 2/20 0.35
RECQL P46063 1/20 0.35
BLM P54132 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
METAP2 P50579 1/20 0.35
LMNA P02545 1/20 0.34
RAB9A P51151 1/20 0.34
MCL1 Q07820 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21075953 0.80 ALDH1A1 (0.43) ALDH1A1STAT3KDM5AAPEX1POLB
SCHEMBL24789857 0.80 OR51E2 (0.37) OR51E2KDM5AMAPTNPSR1
SCHEMBL25014735 0.79 ALDH1A1 (0.44) ALDH1A1STAT3APEX1POLBMEN1
SCHEMBL13618755 0.78 DGAT1 (0.47) ALDH1A1STAT3KDM5AAPEX1POLB
SCHEMBL24050329 0.75 RXFP1 (0.41) ALDH1A1OR51E2POLBMEN1KMT2A
SCHEMBL7523472 0.73 SIGMAR1 (0.44) ALDH1A1POLBMEN1KMT2AMAPT
SCHEMBL10465699 0.72 HSP90AA1 (0.41) ALDH1A1KDM5AMEN1KMT2AMAPT
SCHEMBL25622137 0.71 ALDH1A1 (0.36) ALDH1A1OR51E2STAT3APEX1POLB
SCHEMBL24556716 0.71 ALDH1A1 (0.34) ALDH1A1OR51E2STAT3APEX1POLB
SCHEMBL21558439 0.70 ERN1 (0.53) ALDH1A1POLBKMT2AMAPTKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3666772-A1 DIARYLTHIOHYDANTOIN COMPOUND AS ANDROGEN RECEPTOR ANTAGONIST Chia Tai Tianqing Pharmaceutical Group Co., Ltd. (CN) 2020-06-17 EP disclosed