SCHEMBL13619740

SCHEMBL13619740

N[C@@H](Cc1ccccc1)C(=O)NNC(=O)OCC(=O)NCc1ccccc1

nearest known ligand 0.51

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
MAPT P10636 3/20 0.51
ALDH1A1 P00352 2/20 0.51
HPGD P15428 4/20 0.49
KMT2A Q03164 2/20 0.48
MEN1 O00255 1/20 0.48
TSHR P16473 1/20 0.47
KDM4E B2RXH2 2/20 0.46
CYP1A2 P05177 1/20 0.46
CYP2C9 P11712 1/20 0.46
CYP2C19 P33261 1/20 0.46
GAA P10253 1/20 0.46
LMNA P02545 1/20 0.45
OPRM1 P35372 3/20 0.44
OPRD1 P41143 3/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12371630 0.81 TACR1 (0.64) ALDH1A1
SCHEMBL7413310 0.78 ALPI (0.61) ALDH1A1KMT2A
SCHEMBL3114367 0.78 ALPI (0.61) ALDH1A1KMT2A
SCHEMBL12371604 0.78 CTSS (0.60)
Hydrochloric Acid SCHEMBL27492563 0.76 MMP8 (0.59) ALDH1A1KMT2A
Hydrochloric Acid SCHEMBL3385081 0.76 MMP8 (0.59) ALDH1A1KMT2A
SCHEMBL9364023 0.75 SLC7A5 (0.61) OPRM1OPRD1
SCHEMBL22604490 0.74 CTSS (0.52) OPRM1OPRD1
SCHEMBL10433480 0.73 KMT2A (0.65) MAPTALDH1A1HPGDKMT2AMEN1
SCHEMBL16856328 0.73 PLAU (0.55) KMT2AMEN1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009136997-A2 INHIBITORS OF HUMAN CATHEPSIN L, CATHEPSIN B, AND CATHEPSIN S THE TRUSTEES OF THE UNIVERSITY OF PENNSYLVANIA (US) 2009-11-12 WO disclosed