SCHEMBL13619932

SCHEMBL13619932

COc1cc2c(cc1N)CC(=O)N2

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SRC P12931 2/20 0.46
EGFR P00533 1/20 0.46
EIF2AK2 P19525 1/20 0.44
AHR P35869 4/20 0.41
CMA1 P23946 2/20 0.41
GRIA1 P42261 1/20 0.41
CACNG8 Q8WXS5 1/20 0.41
CCNB2 O95067 1/20 0.40
CDK1 P06493 1/20 0.40
CCNB1 P14635 1/20 0.40
GSK3B P49841 1/20 0.40
CDK5 Q00535 1/20 0.40
CDK5R1 Q15078 1/20 0.40
CCNB3 Q8WWL7 1/20 0.40
S100B P04271 1/20 0.40
PDE3B Q13370 1/20 0.40
PDE3A Q14432 1/20 0.40
ABCB1 P08183 1/20 0.39
L3MBTL1 Q9Y468 2/20 0.39
POLB P06746 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL578508 0.86 SRC (0.57) SRCEGFREIF2AK2AHRCMA1
SCHEMBL28398373 0.85 CYP11B1 (0.52) S100BPDE3BPDE3AL3MBTL1POLB
SCHEMBL21468447 0.83 CYP11B1 (0.44) S100BL3MBTL1POLBCYP19A1CYP11B1
SCHEMBL31335802 0.80 AHR (0.49) SRCEGFREIF2AK2AHRCMA1
SCHEMBL2491904 0.80 AHR (0.50) EIF2AK2AHRCMA1GRIA1CACNG8
SCHEMBL2203230 0.79 CA9 (0.50) S100BPDE3BPDE3AL3MBTL1POLB
SCHEMBL2486755 0.77 GRIA1 (0.51) EIF2AK2AHRCMA1GRIA1CACNG8
SCHEMBL31040248 0.77 AHR (0.49) SRCEGFREIF2AK2AHRCMA1
SCHEMBL5371439 0.77 ACHE (0.46) SRCEGFREIF2AK2AHRCMA1
SCHEMBL2060700 0.76 S100B (0.37) SRCEGFRS100BPDE3BPDE3A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009143389-A1 PHOSPHOROUS DERIVATIVES AS KINASE INHIBITORS ARIAD PHARMACEUTICALS, INC. (US) 2009-11-26 WO disclosed