SCHEMBL13620289

SCHEMBL13620289

CCCCOc1ccc(C[C@H](NC(=O)OC(C)(C)C)C(=O)NNC(=O)SCC(=O)Nc2ccc(C(=O)O)cc2)cc1

nearest known ligand 0.59

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CTSL P07711 4/20 0.59
HDAC8 Q9BY41 1/20 0.51
ITGB3 P05106 1/20 0.48
ITGA2B P08514 1/20 0.48
BCL2 P10415 1/20 0.43
CTSS P25774 4/20 0.42
CTSK P43235 4/20 0.42
HRH2 P25021 3/20 0.42
HRH1 P35367 3/20 0.42
PTPN1 P18031 4/20 0.41
PPARG P37231 1/20 0.40
PPARA Q07869 1/20 0.40
ALDH1A1 P00352 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12372028 0.92 CTSL (0.55) CTSLHDAC8ITGB3ITGA2BBCL2
SCHEMBL12370557 0.84 CTSL (0.81) CTSLHDAC8ITGB3ITGA2BBCL2
SCHEMBL12370592 0.81 CTSL (0.64) CTSLHDAC8ITGB3ITGA2BBCL2
SCHEMBL12371613 0.76 ITGB3 (0.46) CTSLHDAC8ITGB3ITGA2BBCL2
SCHEMBL12371614 0.75 CTSL (0.67) CTSLITGB3ITGA2BBCL2CTSK
SCHEMBL11684068 0.75 CTSS (0.64) CTSLHDAC8ITGB3ITGA2BBCL2
SCHEMBL12372026 0.75 CTSL (0.60) CTSLHDAC8ITGB3ITGA2BBCL2
SCHEMBL12371562 0.75 CTSL (0.50) CTSLHDAC8ITGB3ITGA2BBCL2
SCHEMBL6685168 0.75 ITGB3 (0.79) HDAC8ITGB3ITGA2BPTPN1
SCHEMBL6998950 0.75 ITGB3 (0.79) HDAC8ITGB3ITGA2BPTPN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009136997-A2 INHIBITORS OF HUMAN CATHEPSIN L, CATHEPSIN B, AND CATHEPSIN S THE TRUSTEES OF THE UNIVERSITY OF PENNSYLVANIA (US) 2009-11-12 WO disclosed