SCHEMBL13624018

SCHEMBL13624018

CC(C)C1CC(=O)C=CN1CC(=O)c1ccccc1

nearest known ligand 0.45

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PIK3CD O00329 1/20 0.45
GSK3A P49840 2/20 0.38
GSK3B P49841 2/20 0.38
ALDH1A1 P00352 3/20 0.37
L3MBTL1 Q9Y468 2/20 0.37
HSP90AA1 P07900 1/20 0.37
SMN1; SMN2 Q16637 2/20 0.37
LMNA P02545 1/20 0.37
MAPT P10636 1/20 0.37
HPGD P15428 1/20 0.37
RAB9A P51151 1/20 0.36
NFKB1 P19838 1/20 0.36
NFKB2 Q00653 1/20 0.36
RELA Q04206 1/20 0.36
P2RX7 Q99572 4/20 0.36
DAO P14920 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10200297 0.82 ALDH1A1 (0.42) GSK3AGSK3BALDH1A1L3MBTL1SMN1; SMN2
SCHEMBL13623996 0.80 P2RX7 (0.45) GSK3AGSK3BALDH1A1SMN1; SMN2HPGD
SCHEMBL13624017 0.77 KMT2A (0.40) GSK3AGSK3BALDH1A1L3MBTL1SMN1; SMN2
SCHEMBL13624040 0.72 GRIN2B (0.48) RAB9AP2RX7
SCHEMBL13624015 0.72 ALDH1A1 (0.36) GSK3AGSK3BALDH1A1LMNAP2RX7
SCHEMBL13624010 0.71 P2RX7 (0.39) ALDH1A1L3MBTL1LMNAMAPTP2RX7
SCHEMBL12798882 0.70 RAB9A (0.43) PIK3CDGSK3AGSK3BALDH1A1L3MBTL1
SCHEMBL13624016 0.70 P2RX7 (0.43) ALDH1A1L3MBTL1SMN1; SMN2MAPTHPGD
SCHEMBL3950503 0.65 ALDH1A1 (0.33) PIK3CDALDH1A1SMN1; SMN2P2RX7
SCHEMBL10200295 0.64 ALDH1A1 (0.40) GSK3AGSK3BALDH1A1L3MBTL1HSP90AA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7622489-B2 Kinesin spindle protein inhibitor; antiproliferative agents; anticancer agents; 4-(2,5-difluorophenyl)-N-3-fluoropyrrolidin-3-yl)-2-hydroxymethyl-2-phenyl-2,5-dihydro-1N-pyrrol-1-carboxamide MERCK & CO., INC. (US) 2009-11-24 US disclosed