SCHEMBL13624892

SCHEMBL13624892

Bc1ccc([C@H](C)NCCC(O)(CC(=C)C)c2ccccc2F)cc1

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CNR1 P21554 1/20 0.34
LMNA P02545 3/20 0.32
CYP3A4 P08684 2/20 0.32
CHRM2 P08172 1/20 0.32
HTR1A P08908 1/20 0.32
ADRA2A P08913 1/20 0.32
ADORA3 P0DMS8 1/20 0.32
CHRM1 P11229 1/20 0.32
SMPD1 P17405 1/20 0.32
DRD1 P21728 1/20 0.32
TBXA2R P21731 1/20 0.32
SLC6A2 P23975 1/20 0.32
SLC6A4 P31645 1/20 0.32
ADRA1A P35348 1/20 0.32
OPRM1 P35372 1/20 0.32
DRD3 P35462 1/20 0.32
CASR P41180 1/20 0.32
HTR2B P41595 1/20 0.32
SLC6A3 Q01959 1/20 0.32
KCNH2 Q12809 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL116840 0.90 CNR1 (0.35) CNR1LMNACYP3A4CHRM2HTR1A
SCHEMBL116841 0.90 CNR1 (0.35) CNR1LMNACYP3A4CHRM2HTR1A
SCHEMBL13552217 0.90 HTR1A (0.37) CNR1LMNACYP3A4CHRM2HTR1A
SCHEMBL13552219 0.77 CYP3A4 (0.32) LMNACYP3A4CHRM2HTR1AADRA2A
SCHEMBL117417 0.75 SMN1; SMN2 (0.40) LMNACYP3A4CHRM2HTR1AADRA2A
SCHEMBL13953706 0.69 CYP3A4 (0.38) LMNACYP3A4CHRM2HTR1AADRA2A
SCHEMBL3192627 0.68 SIGMAR1 (0.39) CNR1LMNACYP3A4CHRM2HTR1A
SCHEMBL2698655 0.67 SMN1; SMN2 (0.33) LMNACYP3A4CHRM2HTR1AADRA2A
SCHEMBL734950 0.67 SMN1; SMN2 (0.33) LMNACYP3A4CHRM2HTR1AADRA2A
SCHEMBL1902599 0.65 SMN1; SMN2 (0.43) LMNACYP3A4CHRM2HTR1AADRA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009134400-A1 CYCLIC INHIBITORS OF 11BETA-HYDROXYSTEROID DEHYDROGENASE 1 VITAE PHARMACEUTICALS, INC. (US) 2009-11-05 WO disclosed