SCHEMBL13953706

SCHEMBL13953706

Bc1ccc([C@H](C)NCCC(O)(COC)c2ccccc2)cc1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 2/20 0.38
LMNA P02545 2/20 0.38
OPRM1 P35372 2/20 0.38
HTR1A P08908 2/20 0.38
CHRM2 P08172 1/20 0.38
ADRA2A P08913 1/20 0.38
ADORA3 P0DMS8 1/20 0.38
CHRM1 P11229 1/20 0.38
SMPD1 P17405 1/20 0.38
DRD1 P21728 1/20 0.38
TBXA2R P21731 1/20 0.38
SLC6A2 P23975 1/20 0.38
SLC6A4 P31645 1/20 0.38
ADRA1A P35348 1/20 0.38
DRD3 P35462 1/20 0.38
CASR P41180 1/20 0.38
HTR2B P41595 1/20 0.38
SLC6A3 Q01959 1/20 0.38
KCNH2 Q12809 1/20 0.38
CYP1A2 P05177 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3264659 0.88 LMNA (0.40) CYP3A4LMNAOPRM1HTR1ACHRM2
SCHEMBL118040 0.88 LMNA (0.40) CYP3A4LMNAOPRM1HTR1ACHRM2
SCHEMBL16791656 0.73 SMN1; SMN2 (0.42) CYP3A4LMNAOPRM1HTR1ACHRM2
SCHEMBL10066477 0.72 SMN1; SMN2 (0.40) CYP3A4LMNAOPRM1HTR1ACHRM2
SCHEMBL117417 0.72 SMN1; SMN2 (0.40) CYP3A4LMNAOPRM1HTR1ACHRM2
SCHEMBL15674698 0.72 SMN1; SMN2 (0.40) CYP3A4LMNAOPRM1HTR1ACHRM2
SCHEMBL1692344 0.71 KCNN4 (0.43) KCNH2CYP1A2CYP2C19ALOX15SMN1; SMN2
SCHEMBL15959025 0.70 CYP3A4 (0.53) CYP3A4LMNAOPRM1HTR1ACHRM2
SCHEMBL13624892 0.69 CNR1 (0.34) CYP3A4LMNAOPRM1HTR1ACHRM2
SCHEMBL2065865 0.68 APAF1 (0.43) CYP3A4LMNAOPRM1HTR1ACHRM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009017664-A1 CYCLIC INHIBITORS OF 11β-HYDROXYSTERIOD DEHYDROGENASE 1 VITAE PHARMACEUTICALS, INC. (US) 2009-02-05 WO disclosed