SCHEMBL13625877

SCHEMBL13625877

CCCCc1nc(COC)[nH]c(=O)c1CC1=CC=C(c2ccccc2C#N)CC1

nearest known ligand 0.36

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
APLNR P35414 1/20 0.33
PARP1 P09874 1/20 0.32
ACHE P22303 1/20 0.32
AGTR1 P30556 1/20 0.32
KDM4E B2RXH2 1/20 0.30
ALDH1A1 P00352 1/20 0.30
HPGD P15428 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1891151 0.81 ACHE (0.43) APLNRACHEAGTR1
SCHEMBL13626562 0.79
SCHEMBL27771424 0.76 CYP19A1 (0.37) APLNRPARP1ACHEKDM4EALDH1A1
SCHEMBL13625909 0.75 ACHE (0.34) APLNRACHEAGTR1
SCHEMBL1889439 0.74 ACHE (0.42) APLNRACHEAGTR1
SCHEMBL3487184 0.73 PARP1 (0.38) APLNRPARP1ACHEAGTR1
SCHEMBL13626516 0.73 AGTR1 (0.33) APLNRACHEAGTR1KDM4EALDH1A1
SCHEMBL12348665 0.72 ACHE (0.45) APLNRACHEAGTR1
SCHEMBL1894561 0.72 ACHE (0.45) APLNRPARP1ACHEAGTR1
SCHEMBL1886429 0.71 ACHE (0.43) PARP1ACHEAGTR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009133970-A1 CRYSTALLINE COMPOUND TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2009-11-05 WO disclosed