SCHEMBL13626185

SCHEMBL13626185

CCc1sc(C(=O)Nc2cc(-c3ccnc(Nc4ccc(N5CCN(C)CC5)cc4)n3)ccc2F)cc1C(C)C

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
JAK2 O60674 8/20 0.53
JAK3 P52333 3/20 0.49
HDAC1 Q13547 1/20 0.49
HDAC6 Q9UBN7 1/20 0.49
EGFR P00533 4/20 0.47
STK17A Q9UEE5 1/20 0.45
KIT P10721 2/20 0.45
ERBB2 P04626 2/20 0.45
IGF1R P08069 2/20 0.45
IKBKB O14920 1/20 0.45
CHUK O15111 1/20 0.45
PLK4 O00444 1/20 0.45
CHEK1 O14757 1/20 0.45
AURKA O14965 1/20 0.45
DAPK3 O43293 1/20 0.45
ROCK2 O75116 1/20 0.45
PRKD3 O94806 1/20 0.45
MAP4K4 O95819 1/20 0.45
PAK4 O96013 1/20 0.45
CHEK2 O96017 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13626485 0.85 SYK (0.47) JAK2AURKANTRK1ROS1FLT3
SCHEMBL1422805 0.81 JAK2 (0.53) JAK2JAK3HDAC1HDAC6EGFR
SCHEMBL13626131 0.76 BTK (0.43) EGFRBTK
SCHEMBL13626133 0.75 BTK (0.57) BTK
SCHEMBL13626128 0.74 BTK (0.41) EGFRBTK
SCHEMBL13626828 0.74 BTK (0.43) EGFRNTRK1METSRCBTK
SCHEMBL13626122 0.73 BTK (0.55) BTK
SCHEMBL13626829 0.73 BTK (0.55) BTK
SCHEMBL13626182 0.72 BTK (0.48) BTKSLKKCNH2
SCHEMBL13626831 0.71 BTK (0.51) BTK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009137596-A1 SUBSTITUTED AMIDES, METHOD OF MAKING, AND USE AS BTK INHIBITORS CGI PHARMACEUTICALS, INC. (US) 2009-11-12 WO disclosed