SCHEMBL13626817

SCHEMBL13626817

C[C@@H](CO)COc1cccc(C(=O)Nc2cccc3ccc(-c4cccc(C(F)(F)F)c4)nc23)c1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TP53 P04637 1/20 0.48
POLB P06746 1/20 0.48
ALDH1A1 P00352 2/20 0.44
THRB P10828 1/20 0.44
RXFP1 Q9HBX9 3/20 0.42
GAA P10253 2/20 0.41
CYP1A2 P05177 1/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2D6 P10635 1/20 0.41
CYP2C19 P33261 1/20 0.41
PLG P00747 1/20 0.41
PLAU P00749 1/20 0.41
PLAT P00750 1/20 0.41
TRPV3 Q8NET8 1/20 0.40
GPR52 Q9Y2T5 1/20 0.40
NPSR1 Q6W5P4 2/20 0.39
MAPT P10636 2/20 0.39
CNR2 P34972 1/20 0.39
MAPK1 P28482 1/20 0.39
TDP1 Q9NUW8 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1034692 0.92 TP53 (0.47) TP53POLBALDH1A1THRBRXFP1
SCHEMBL1034693 0.92 TP53 (0.47) TP53POLBALDH1A1THRBRXFP1
SCHEMBL1034276 0.85 THRB (0.58) TP53POLBALDH1A1THRBRXFP1
SCHEMBL13627127 0.81 PLG (0.45) RXFP1PLGPLAUPLATTRPV3
SCHEMBL1034348 0.79 EPHX2 (0.52) TP53POLBRXFP1GAAMAP4K4
SCHEMBL1034793 0.78 ALDH1A1 (0.48) TP53ALDH1A1RXFP1GAAPLG
SCHEMBL1035268 0.78 GPR52 (0.44) ALDH1A1GAATRPV3GPR52MAPT
SCHEMBL1035266 0.78 GPR52 (0.44) ALDH1A1GAATRPV3GPR52MAPT
SCHEMBL1035575 0.76 RXFP1 (0.44) RXFP1PLGPLAUPLATMAPT
SCHEMBL1032642 0.76 RXFP1 (0.44) RXFP1PLGPLAUPLATMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009134973-A1 QUENOLINES AND RELATED ANALOGS AS SIRTUIN MODULATORS SIRTRIS PHARMACEUTICALS, INC. (US) 2009-11-05 WO disclosed