SCHEMBL13627327

SCHEMBL13627327

Cc1cc(-c2ccccc2C(F)(F)F)cc2c1NC[C@H]1CNC[C@@H]21

nearest known ligand 0.42

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
TRPA1 O75762 3/20 0.42
HTR2A P28223 8/20 0.36
HTR2C P28335 8/20 0.36
HTR2B P41595 8/20 0.36
TRPM8 Q7Z2W7 1/20 0.34
TRPV1 Q8NER1 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4478989 1.00 TRPA1 (0.42) TRPA1HTR2AHTR2CHTR2BTRPM8
SCHEMBL4482328 1.00 TRPA1 (0.42) TRPA1HTR2AHTR2CHTR2BTRPM8
SCHEMBL13627313 0.86 TRPA1 (0.36) TRPA1HTR2AHTR2CHTR2BTRPM8
SCHEMBL4477342 0.86 TRPA1 (0.36) TRPA1HTR2AHTR2CHTR2BTRPM8
SCHEMBL4472523 0.86 TRPA1 (0.36) TRPA1HTR2AHTR2CHTR2BTRPM8
SCHEMBL4483043 0.80 HTR2C (0.33) HTR2AHTR2CHTR2B
SCHEMBL13627326 0.80 HTR2C (0.33) HTR2AHTR2CHTR2B
SCHEMBL13627348 0.80 TRPA1 (0.41) TRPA1HTR2AHTR2CHTR2BTRPM8
SCHEMBL4477738 0.80 TRPA1 (0.41) TRPA1HTR2AHTR2CHTR2BTRPM8
SCHEMBL13627329 0.74 HTR2C (0.42) HTR2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7618980-B2 Pyrrolo(oxo)quinolines as 5HT ligands BRISTOL-MYERS SQUIBB COMPANY (US) 2009-11-17 US disclosed