SCHEMBL13627330

SCHEMBL13627330

Cc1cc(Nc2ccccc2)cc2c1N(C)C[C@H]1CNC[C@@H]21

nearest known ligand 0.33

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
BPTF Q12830 1/20 0.33
OPRM1 P35372 1/20 0.32
OPRD1 P41143 1/20 0.32
OPRK1 P41145 1/20 0.32
APP P05067 1/20 0.32
NPSR1 Q6W5P4 1/20 0.31
HPGD P15428 1/20 0.30
CHRNB4 P30926 1/20 0.30
CHRNA3 P32297 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4472029 1.00 BPTF (0.33) BPTFOPRM1OPRD1OPRK1APP
SCHEMBL4482834 0.85 BRAF (0.34) BPTFOPRM1OPRD1OPRK1APP
SCHEMBL13627342 0.85 BRAF (0.34) BPTFOPRM1OPRD1OPRK1APP
SCHEMBL4492625 0.84 CHRNB2 (0.40) OPRM1OPRD1OPRK1HPGDCHRNB4
SCHEMBL13627337 0.84 CHRNB2 (0.40) OPRM1OPRD1OPRK1HPGDCHRNB4
SCHEMBL13627331 0.83 HTR2A (0.35) NPSR1
SCHEMBL4472375 0.83 HTR2A (0.35) NPSR1
SCHEMBL4472041 0.83 HTR2A (0.35) NPSR1
SCHEMBL4489439 0.80 HTR2C (0.38)
SCHEMBL13627333 0.80 HTR2C (0.38)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7618980-B2 Pyrrolo(oxo)quinolines as 5HT ligands BRISTOL-MYERS SQUIBB COMPANY (US) 2009-11-17 US disclosed