SCHEMBL13633239

SCHEMBL13633239

COc1cccc(C2CC(=O)C=CN2C(=O)OCc2ccccc2)c1

nearest known ligand 0.48

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 6/20 0.48
ALDH1A1 P00352 1/20 0.44
LMNA P02545 1/20 0.43
MAPT P10636 1/20 0.43
HTT P42858 1/20 0.43
TMEM97 Q5BJF2 3/20 0.42
SIGMAR1 Q99720 3/20 0.42
NPSR1 Q6W5P4 1/20 0.42
BCL9 O00512 1/20 0.42
CTNNB1 P35222 1/20 0.42
TP53 P04637 1/20 0.42
FABP7 O15540 1/20 0.40
FABP5 Q01469 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20449200 0.87 P2RX7 (0.49) P2RX7TMEM97SIGMAR1NPSR1FABP7
SCHEMBL3159251 0.87 P2RX7 (0.49) P2RX7TMEM97SIGMAR1NPSR1FABP7
SCHEMBL20703481 0.85 PKM (0.47) P2RX7ALDH1A1LMNATMEM97SIGMAR1
SCHEMBL13634012 0.84 P2RX7 (0.45) P2RX7ALDH1A1MAPTHTTTMEM97
SCHEMBL2724266 0.82 P2RX7 (0.42) P2RX7MAPTHTTTMEM97SIGMAR1
SCHEMBL31462845 0.81 MAPT (0.47) P2RX7ALDH1A1MAPTHTTTMEM97
SCHEMBL2706680 0.80 P2RX7 (0.47) P2RX7TMEM97SIGMAR1FABP7FABP5
SCHEMBL3167642 0.79 PTGDR2 (0.44) P2RX7
SCHEMBL13634008 0.79 MITF (0.40) P2RX7MAPTHTT
SCHEMBL13624040 0.78 GRIN2B (0.48) P2RX7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7622489-B2 Kinesin spindle protein inhibitor; antiproliferative agents; anticancer agents; 4-(2,5-difluorophenyl)-N-3-fluoropyrrolidin-3-yl)-2-hydroxymethyl-2-phenyl-2,5-dihydro-1N-pyrrol-1-carboxamide MERCK & CO., INC. (US) 2009-11-24 US disclosed