SCHEMBL13633552

SCHEMBL13633552

O=C(O)c1cn2c(Cl)cc(-c3cccnc3)cc2n1

nearest known ligand 0.45

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
KMO O15229 2/20 0.45
MKNK1 Q9BUB5 4/20 0.43
MKNK2 Q9HBH9 4/20 0.43
PIM1 P11309 1/20 0.43
PIM2 Q9P1W9 1/20 0.43
CYP19A1 P11511 1/20 0.41
GLO1 Q04760 1/20 0.40
NR4A2 P43354 1/20 0.39
DHODH Q02127 1/20 0.39
CSNK2A2 P19784 1/20 0.39
CSNK2B P67870 1/20 0.39
CSNK2A1 P68400 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13633542 0.83 GAA (0.50)
SCHEMBL13633515 0.74 MAP3K5 (0.44)
SCHEMBL13633503 0.71 GAA (0.50)
SCHEMBL1282214 0.71 RXFP1 (0.41) DHODH
SCHEMBL119204 0.70 PTGS1 (0.51)
SCHEMBL23455357 0.69 MKNK1 (0.57) KMOMKNK1MKNK2PIM1PIM2
SCHEMBL30073951 0.69 MKNK1 (0.57) KMOMKNK1MKNK2PIM1PIM2
SCHEMBL4778479 0.69 KMO (0.53) KMOMKNK1MKNK2PIM1PIM2
SCHEMBL3262905 0.69 ALDH1A1 (0.49) MKNK1MKNK2CYP19A1
SCHEMBL21713059 0.68 KMO (0.48) KMOMKNK1MKNK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20090275577-A1 IMIDAZOPYRIDINE AND IMIDAZOPYRIMIDINE DERIVATIVES AS ANTIBACTERIAL AGENTS PFIZER INC 2009-11-05 US disclosed
US-7563788-B2 Substituted Imidazo[1,2-a]pyridines as Antibacterial Agents PFIZER INC. (US) 2009-07-21 US disclosed
US-7563788-B2 Substituted Imidazo[1,2-a]pyridines as Antibacterial Agents PFIZER INC. (US) 2009-07-21 US disclosed
US-20070191394-A1 Antibacterial agents WARNER-LAMBERT COMPANY LLC 2007-08-16 US disclosed
US-20070191394-A1 Antibacterial agents WARNER-LAMBERT COMPANY LLC 2007-08-16 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070191394-A1 Antibacterial agents MRPL21, RPN2, FBL KMO 4218/4885MKNK1 2780/4885MKNK2 2662/4885
US-20090275577-A1 IMIDAZOPYRIDINE AND IMIDAZOPYRIMIDINE DERIVATIVES AS ANTIBACTERIAL AGENTS DPYD, TYMP, ITPA KMO 4206/4885MKNK1 2093/4885MKNK2 2022/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.