SCHEMBL13634124

SCHEMBL13634124

CCn1c2ccccc2c2cc(N(c3ccccc3)c3ccc4c(c3)C3(c5ccccc5-c5ccccc53)c3ccccc3-4)ccc21

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 6/20 0.45
KDM4E B2RXH2 5/20 0.45
MEN1 O00255 4/20 0.45
KMT2A Q03164 4/20 0.45
MAPK1 P28482 3/20 0.45
TDP1 Q9NUW8 2/20 0.45
HTT P42858 2/20 0.45
ALDH1A1 P00352 2/20 0.45
HPGD P15428 1/20 0.45
HBB P68871 1/20 0.45
HSD17B10 Q99714 1/20 0.45
LMNA P02545 4/20 0.41
NPY5R Q15761 2/20 0.41
POLB P06746 3/20 0.40
BLM P54132 1/20 0.40
PKM P14618 1/20 0.40
RORC P51449 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
DRD3 P35462 1/20 0.39
SRC P12931 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24022276 0.96 MAPT (0.48) MAPTKDM4EMEN1KMT2AMAPK1
SCHEMBL24022285 0.93 KDM1A (0.40) MAPTKDM4EMEN1KMT2AMAPK1
SCHEMBL13803219 0.92 TSPO (0.44) MAPTKDM4EMEN1KMT2AMAPK1
SCHEMBL21940003 0.91 RORC (0.36) MAPTKDM4EMEN1KMT2AMAPK1
SCHEMBL13634132 0.91 ALDH1A1 (0.46) MAPTKDM4EMEN1KMT2AMAPK1
SCHEMBL21984811 0.90 MAPT (0.41) MAPTKDM4EMEN1KMT2AMAPK1
SCHEMBL24022286 0.90 MAPT (0.45) MAPTKDM4EMEN1KMT2AMAPK1
SCHEMBL24022110 0.90 TSPO (0.39) MAPTKDM4EMEN1KMT2AMAPK1
SCHEMBL14466303 0.89 MAPT (0.46) MAPTKDM4EMEN1KMT2AMAPK1
SCHEMBL21940170 0.89 KDM1A (0.42) MAPTKDM4EMEN1KMT2AMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 16 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20180175295-A1 SPIROFLUORENE DERIVATIVE, MATERIAL FOR LIGHT-EMITTING ELEMENT, LIGHT-EMITTING ELEMENT, LIGHT-EMITTING DEVICE, AND ELECTRONIC DEVICE SEMICONDUCTOR ENERGY LAB (JP) 2018-06-21 US disclosed
US-9899602-B2 Spirofluorene derivative, material for light-emitting element, light-emitting element, light-emitting device, and electronic device SEMICONDUCTOR ENERGY LABORATORY CO., LTD. (JP) 2018-02-20 US disclosed
US-20170125679-A1 SPIROFLUORENE DERIVATIVE, MATERIAL FOR LIGHT-EMITTING ELEMENT, LIGHT-EMITTING ELEMENT, LIGHT-EMITTING DEVICE, AND ELECTRONIC DEVICE SEMICONDUCTOR ENERGY LAB (JP) 2017-05-04 US disclosed
US-9548457-B2 Spirofluorene derivative, material for light-emitting element, light-emitting element, light-emitting device, and electronic device SEMICONDUCTOR ENERGY LABORATORIES CO., LTD. (JP) 2017-01-17 US disclosed
US-9548457-B2 Spirofluorene derivative, material for light-emitting element, light-emitting element, light-emitting device, and electronic device SEMICONDUCTOR ENERGY LABORATORIES CO., LTD. (JP) 2017-01-17 US disclosed
US-20160087209-A1 SPIROFLUORENE DERIVATIVE, MATERIAL FOR LIGHT-EMITTING ELEMENT, LIGHT-EMITTING ELEMENT, LIGHT-EMITTING DEVICE, AND ELECTRONIC DEVICE SEMICONDUCTOR ENERGY LAB (JP) 2016-03-24 US disclosed
US-20160087209-A1 SPIROFLUORENE DERIVATIVE, MATERIAL FOR LIGHT-EMITTING ELEMENT, LIGHT-EMITTING ELEMENT, LIGHT-EMITTING DEVICE, AND ELECTRONIC DEVICE SEMICONDUCTOR ENERGY LAB (JP) 2016-03-24 US disclosed
US-9203035-B2 Spirofluorene derivative, material for light-emitting element, light-emitting element, light-emitting device, and electronic device SEMICONDUCTOR ENERGY LABORATORY CO., LTD. (KE) 2015-12-01 US disclosed
US-20140213798-A1 SPIROFLUORENE DERIVATIVE, MATERIAL FOR LIGHT-EMITTING ELEMENT, LIGHT-EMITTING ELEMENT, LIGHT-EMITTING DEVICE, AND ELECTRONIC DEVICE SEMICONDUCTOR ENERGY LABORATORY CO., LTD. (JP) 2014-07-31 US disclosed
US-8704212-B2 Spirofluorene derivative, material for light-emitting element, light-emitting element, light-emitting device, and electronic device SEMICONDUCTOR ENERGY LABORATORY CO., LTD. (JP) 2014-04-22 US disclosed
US-8304094-B2 High light efficincy; hole transporting substance; phosphorescence SEMICONDUCTOR ENERGY LABORATORY CO., LTD. (JP) 2012-11-06 US disclosed
US-8304094-B2 High light efficincy; hole transporting substance; phosphorescence SEMICONDUCTOR ENERGY LABORATORY CO., LTD. (JP) 2012-11-06 US disclosed
WO-2008105349-A1 LIGHT-EMITTING ELEMENT USING SPIROFLUORENE DERIVATIVE AND ELECTRONIC APPLIANCE SEMICONDUCTOR ENERGY LABORATORY CO., LTD. (JP) 2008-09-04 WO disclosed
US-20080206598-A1 Light-emitting element using spirofluorene derivative and electronic appliance SEMICONDUCTOR ENERGY LABORATORY CO., LTD. (JP) 2008-08-28 US disclosed
US-20080206598-A1 Light-emitting element using spirofluorene derivative and electronic appliance SEMICONDUCTOR ENERGY LABORATORY CO., LTD. (JP) 2008-08-28 US disclosed
WO-2007043354-A9 SPIROFLUORENE DERIVATIVE, MATERIAL FOR LIGHT-EMITTING ELEMENT, LIGHT-EMITTING ELEMENT, LIGHT-EMITTING DEVICE, AND ELECTRONIC DEVICE SEMICONDUCTOR ENERGY LAB (JP) 2007-06-07 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20170125679-A1 SPIROFLUORENE DERIVATIVE, MATERIAL FOR LIGHT-EMITTING ELEMENT, LIGHT-EMITTING ELEMENT, LIGHT-EMITTING DEVICE, AND ELECTRONIC DEVICE GRK1, PTGER2, PTGER1 MAPT 4329/4885KDM4E 4076/4885MEN1 2313/4885
US-20180175295-A1 SPIROFLUORENE DERIVATIVE, MATERIAL FOR LIGHT-EMITTING ELEMENT, LIGHT-EMITTING ELEMENT, LIGHT-EMITTING DEVICE, AND ELECTRONIC DEVICE GRK1, PTGER2, PTGER1 MAPT 4329/4885KDM4E 4076/4885MEN1 2313/4885
US-20160087209-A1 SPIROFLUORENE DERIVATIVE, MATERIAL FOR LIGHT-EMITTING ELEMENT, LIGHT-EMITTING ELEMENT, LIGHT-EMITTING DEVICE, AND ELECTRONIC DEVICE GRK1, PTGER2, PTGER1 MAPT 4329/4885KDM4E 4076/4885MEN1 2313/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.