SCHEMBL13634686

SCHEMBL13634686

COC[C@H]1CCCN1Cc1ccc(NC(=O)c2csc(Br)n2)c(C(=O)NC2CCOCC2)c1

nearest known ligand 0.47

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
HDAC8 Q9BY41 2/20 0.47
HDAC6 Q9UBN7 2/20 0.47
HDAC1 Q13547 1/20 0.47
S1PR1 P21453 1/20 0.45
PIM1 P11309 2/20 0.40
MCHR1 Q99705 3/20 0.38
PDE4B Q07343 1/20 0.37
SMYD3 Q9H7B4 1/20 0.37
IRAK4 Q9NWZ3 1/20 0.37
P2RX7 Q99572 1/20 0.36
SIGMAR1 Q99720 2/20 0.36
ADORA2A P29274 1/20 0.35
ADORA1 P30542 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13634853 0.89 HDAC8 (0.42) HDAC8HDAC6HDAC1S1PR1PIM1
SCHEMBL13162967 0.88 HDAC8 (0.50) HDAC8HDAC6HDAC1S1PR1SIGMAR1
SCHEMBL13634771 0.87 S1PR1 (0.49) HDAC8HDAC6HDAC1S1PR1SIGMAR1
SCHEMBL13634649 0.87 S1PR1 (0.42) HDAC8HDAC6HDAC1S1PR1PIM1
SCHEMBL13270431 0.81 S1PR1 (0.38) HDAC8HDAC6HDAC1S1PR1PIM1
SCHEMBL15888674 0.81 S1PR1 (0.38) HDAC8HDAC6HDAC1S1PR1PIM1
SCHEMBL13638887 0.80 S1PR1 (0.47) HDAC8HDAC6HDAC1S1PR1IRAK4
SCHEMBL13270753 0.80 HDAC8 (0.54) HDAC8HDAC6HDAC1S1PR1MCHR1
SCHEMBL13634841 0.80 S1PR1 (0.49) HDAC8HDAC6HDAC1S1PR1IRAK4
SCHEMBL13163118 0.79 HDAC8 (0.53) HDAC8HDAC6HDAC1S1PR1MCHR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8304547-B2 Azolecarboxamide compound or salt thereof ASTELLAS PHARMA INC. (JP) 2012-11-06 US disclosed
US-8304547-B2 Azolecarboxamide compound or salt thereof ASTELLAS PHARMA INC. (JP) 2012-11-06 US disclosed