SCHEMBL13634771

SCHEMBL13634771

CCCNC(=O)c1cc(CN2CCC[C@@H]2COC)ccc1NC(=O)c1csc(Br)n1

nearest known ligand 0.49

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 1/20 0.49
HDAC8 Q9BY41 2/20 0.49
HDAC6 Q9UBN7 2/20 0.49
HDAC1 Q13547 1/20 0.49
SIGMAR1 Q99720 2/20 0.40
DRD2 P14416 3/20 0.40
ACKR3 P25106 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13162967 0.95 HDAC8 (0.50) S1PR1HDAC8HDAC6HDAC1SIGMAR1
SCHEMBL13634595 0.88 S1PR1 (0.49) S1PR1HDAC8HDAC6HDAC1SIGMAR1
SCHEMBL13634686 0.87 HDAC8 (0.47) S1PR1HDAC8HDAC6HDAC1SIGMAR1
SCHEMBL13634729 0.87 S1PR1 (0.45) S1PR1HDAC8HDAC6HDAC1SIGMAR1
SCHEMBL13634841 0.84 S1PR1 (0.49) S1PR1HDAC8HDAC6HDAC1SIGMAR1
SCHEMBL13638884 0.83 S1PR1 (0.47) S1PR1HDAC8HDAC6HDAC1SIGMAR1
SCHEMBL13638916 0.82 HDAC8 (0.43) S1PR1HDAC8HDAC6HDAC1SIGMAR1
SCHEMBL13634557 0.80 S1PR1 (0.42) S1PR1HDAC8HDAC6HDAC1SIGMAR1
SCHEMBL13270465 0.80 KMT2A (0.44)
SCHEMBL13638887 0.79 S1PR1 (0.47) S1PR1HDAC8HDAC6HDAC1SIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8304547-B2 Azolecarboxamide compound or salt thereof ASTELLAS PHARMA INC. (JP) 2012-11-06 US disclosed