SCHEMBL13635124

SCHEMBL13635124

O=C(O)c1ccc2c3ccccc3n(C3CCNC3)c2c1

nearest known ligand 0.44

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
KDM2B Q8NHM5 1/20 0.44
KDM4E B2RXH2 2/20 0.44
HTR6 P50406 6/20 0.43
ALDH1A1 P00352 1/20 0.40
HPGD P15428 1/20 0.40
PARP1 P09874 2/20 0.39
KHK P50053 3/20 0.38
PTGER4 P35408 1/20 0.37
SLC6A2 P23975 1/20 0.36
SLC6A4 P31645 1/20 0.36
SLC6A3 Q01959 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13011465 1.00 KDM2B (0.44) KDM2BKDM4EHTR6ALDH1A1HPGD
SCHEMBL13061916 0.92 KDM4E (0.46) KDM2BKDM4EHTR6ALDH1A1HPGD
SCHEMBL13011488 0.86 KIF11 (0.44) HTR6ALDH1A1PARP1PTGER4
SCHEMBL13011487 0.86 KIF11 (0.44) HTR6ALDH1A1PARP1PTGER4
SCHEMBL13011766 0.84 HTR2B (0.46) HTR6SLC6A3
SCHEMBL13011750 0.84 HTR2B (0.46) HTR6SLC6A3
SCHEMBL23697539 0.82 HTR6 (0.49) HTR6KHKSLC6A4
SCHEMBL23697542 0.82 HTR6 (0.49) HTR6KHKSLC6A4
SCHEMBL13061928 0.82 L3MBTL1 (0.51) KDM4EALDH1A1HPGDPARP1
SCHEMBL13011348 0.81 KDM4E (0.47) KDM4EALDH1A1HPGDPARP1PTGER4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2119704-A1 ACYLGUANIDINE DERIVATIVE Astellas Pharma Inc. (JP) 2009-11-18 EP disclosed