SCHEMBL13636880

SCHEMBL13636880

C=C(NC1(C(=O)NCc2cc(C)on2)CC1)c1cc(C(C)(C)C)nc(C(C)(C)C)c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EPHX2 P34913 2/20 0.43
NPC1 O15118 2/20 0.36
RAB9A P51151 2/20 0.36
ADORA2A P29274 1/20 0.36
ADORA1 P30542 1/20 0.36
ROCK2 O75116 1/20 0.34
KMT2A Q03164 1/20 0.34
FPR3 P25089 1/20 0.34
FPR2 P25090 1/20 0.34
HDAC1 Q13547 1/20 0.33
HDAC6 Q9UBN7 1/20 0.33
NAMPT P43490 1/20 0.33
SMN1; SMN2 Q16637 2/20 0.33
MAPK1 P28482 1/20 0.32
CYP3A4 P08684 1/20 0.32
CYP2C9 P11712 1/20 0.32
CYP2C19 P33261 1/20 0.32
PDE10A Q9Y233 1/20 0.32
ALDH1A1 P00352 1/20 0.31
TP53 P04637 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7857531 0.91 EPHX2 (0.44) EPHX2NPC1RAB9AADORA2AADORA1
SCHEMBL7859105 0.87 EPHX2 (0.43) EPHX2NPC1RAB9AADORA2AADORA1
SCHEMBL7859092 0.86 EPHX2 (0.42) EPHX2NPC1RAB9AADORA2AADORA1
SCHEMBL7856656 0.77 EPHX2 (0.43) EPHX2NPC1RAB9AADORA2AADORA1
SCHEMBL7855762 0.76 EPHX2 (0.43) EPHX2KMT2ACYP3A4CYP2C9CYP2C19
SCHEMBL7856605 0.74 P2RX3 (0.39)
SCHEMBL7848736 0.73 EPHX2 (0.41) EPHX2ROCK2CYP3A4CYP2C9CYP2C19
SCHEMBL7857567 0.71 POLB (0.47) NPC1RAB9AKMT2ASMN1; SMN2ALDH1A1
SCHEMBL7856575 0.71 EPHX2 (0.39) EPHX2CYP3A4CYP2C9CYP2C19PDE10A
SCHEMBL13636839 0.70 FPR2 (0.46) NPC1RAB9AKMT2AFPR2SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009132453-A1 CYCLYLAMINE DERIVATIVES AS CALCIUM CHANNEL BLOCKERS NEUROMED PHARMACEUTICALS LTD. (CA) 2009-11-05 WO disclosed