SCHEMBL13637752

SCHEMBL13637752

C[C@@H](C(=O)N[C@@H](CC(=O)O)C(=O)c1ncc(-c2c(Cl)cccc2Cl)o1)n1cccc(NC=O)c1=O

nearest known ligand 0.43

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CASP3 P42574 4/20 0.43
CASP1 P29466 10/20 0.42
CASP7 P55210 1/20 0.42
CASP8 Q14790 1/20 0.42
IL1B P01584 1/20 0.41
ELANE P08246 6/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12450477 0.86 CASP1 (0.57) CASP3CASP1CASP7CASP8IL1B
SCHEMBL473286 0.67 CASP1 (0.56) CASP3CASP1CASP8IL1BELANE
SCHEMBL473285 0.67 CASP1 (0.56) CASP3CASP1CASP8IL1BELANE
SCHEMBL12946365 0.67 CASP3 (0.46) CASP3
SCHEMBL12946449 0.66 CASP1 (0.51) CASP3CASP1CASP7
SCHEMBL12450478 0.66 CASP1 (0.58) CASP3CASP1IL1BELANE
SCHEMBL12450469 0.65 CASP1 (0.58) CASP3CASP1CASP7CASP8IL1B
SCHEMBL12450525 0.64 CASP3 (0.40) CASP3CASP1IL1B
SCHEMBL13637689 0.64 CASP1 (0.42) CASP3CASP1CASP8IL1B
SCHEMBL473088 0.62 CASP1 (0.55) CASP3CASP1CASP7CASP8IL1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2123665-A2 Inhibitors of interleukin-1Beta converting enzyme Vertex Pharmaceuticals Incorporated (US) 2009-11-25 EP disclosed