SCHEMBL13637770

SCHEMBL13637770

CS(=O)(=O)c1ccc2c(c1)cc(C1CC=C(C(=O)O)O1)n2Cc1ccc(F)cc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCR2 P41597 2/20 0.48
PTGS2 P35354 6/20 0.45
TBXA2R P21731 3/20 0.41
PTGDR Q13258 2/20 0.38
PTGDR2 Q9Y5Y4 1/20 0.37
SERPINE1 P05121 1/20 0.36
GNRHR P30968 2/20 0.36
MEN1 O00255 1/20 0.36
ALDH1A1 P00352 1/20 0.36
CYP3A4 P08684 1/20 0.36
MAPT P10636 1/20 0.36
CYP2C9 P11712 1/20 0.36
HPGD P15428 1/20 0.36
MAPK1 P28482 1/20 0.36
CYP2C19 P33261 1/20 0.36
KMT2A Q03164 1/20 0.36
HSD17B10 Q99714 1/20 0.36
PTGS1 P23219 2/20 0.35
AGTR1 P30556 1/20 0.35
AGTR2 P50052 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2921656 0.80 PTGS2 (0.48) CCR2PTGS2TBXA2RPTGDRGNRHR
SCHEMBL2924383 0.78 CCR2 (0.76) CCR2PTGS2TBXA2RSERPINE1
SCHEMBL2920935 0.77 PTGS2 (0.49) CCR2PTGS2TBXA2RPTGDRGNRHR
SCHEMBL2920685 0.74 PTGS2 (0.56) CCR2PTGS2TBXA2RPTGDR2
SCHEMBL2927892 0.73 PTGS2 (0.61) CCR2PTGS2TBXA2RPTGDR2SERPINE1
SCHEMBL2925670 0.72 CCR2 (0.51) CCR2PTGS2TBXA2RPTGDR2SERPINE1
SCHEMBL2929127 0.72 PTGS2 (0.56) CCR2PTGS2TBXA2RPTGDR2GNRHR
SCHEMBL2929297 0.71 PTGS2 (0.82) CCR2PTGS2TBXA2RALDH1A1MAPT
SCHEMBL8069895 0.71 PTGS2 (0.56) CCR2PTGS2TBXA2RALDH1A1CYP3A4
SCHEMBL2923938 0.70 PTGS2 (0.56) CCR2PTGS2TBXA2RPTGDR2GNRHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7612070-B2 Heterocyclic compounds as antiinflammatory agents and cyclooxygenase inhibitors CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2009-11-03 US disclosed