SCHEMBL13658809

SCHEMBL13658809

NC(=O)c1cccc2cc(NS(=O)(=O)c3cc(Cl)cc(I)c3)ccc12

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2C9 P11712 1/20 0.43
ATIC P31939 1/20 0.43
CYP2C19 P33261 1/20 0.43
HSD17B10 Q99714 1/20 0.43
MEN1 O00255 1/20 0.42
KMT2A Q03164 1/20 0.42
ACLY P53396 1/20 0.41
MAPK1 P28482 1/20 0.40
KDM4E B2RXH2 1/20 0.39
ALDH1A1 P00352 1/20 0.39
GAA P10253 1/20 0.39
CASP1 P29466 1/20 0.39
HSP90AA1 P07900 1/20 0.39
HSP90AB1 P08238 1/20 0.39
PGR P06401 2/20 0.39
AKR1C3 P42330 1/20 0.39
PKM P14618 1/20 0.39
HTR6 P50406 1/20 0.39
CYP19A1 P11511 1/20 0.39
GPR27 Q9NS67 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1110383 0.92 ACLY (0.48) CYP2C9ATICCYP2C19HSD17B10MEN1
SCHEMBL1110258 0.82 ACLY (0.58) CYP2C9ATICCYP2C19HSD17B10MEN1
SCHEMBL1110309 0.82 ACLY (0.49) CYP2C9ATICCYP2C19HSD17B10ACLY
SCHEMBL13658789 0.80 CHEK2 (0.45) ATICALDH1A1GAAPGRAKR1C3
SCHEMBL1320440 0.79 ACLY (0.49) CYP2C9ATICCYP2C19HSD17B10ACLY
SCHEMBL13658687 0.76 TUBB (0.41) MEN1KMT2A
SCHEMBL13658722 0.75 CYP2C9 (0.60) CYP2C9ATICCYP2C19HSD17B10ACLY
SCHEMBL1320525 0.74 KCNA5 (0.52) MEN1KMT2AACLYALDH1A1PGR
SCHEMBL13905620 0.74 TUBB (0.48) CYP2C9ATICCYP2C19HSD17B10MEN1
SCHEMBL1110473 0.73 PGR (0.47) CYP2C9ATICCYP2C19HSD17B10MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009127723-A1 NEW ARYLSULPHONYLGLYCINE DERIVATIVES, THE PREPARATION THEREOF AND THEIR USE AS MEDICAMENTS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2009-10-22 WO disclosed