SCHEMBL13660413

SCHEMBL13660413

Cc1csc2c(=O)n(-c3ccc(C#N)nc3)c([C@H]3C[C@@H]4[C@H](C3)C4(F)F)nc12

nearest known ligand 0.34

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
DPP4 P27487 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.32
USP14 P54578 2/20 0.31
PDE4B Q07343 2/20 0.31
PDE4D Q08499 1/20 0.31
PDE7A Q13946 1/20 0.31
GRM1 Q13255 1/20 0.30
OPRM1 P35372 1/20 0.30
OPRL1 P41146 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13660457 0.88 DPP4 (0.34) DPP4SMN1; SMN2PDE4BPDE7A
SCHEMBL13660414 0.87 SMN1; SMN2 (0.34) SMN1; SMN2PDE4BPDE7AGRM1
SCHEMBL13985419 0.78 PDE4B (0.34) DPP4USP14PDE4BPDE4DOPRM1
SCHEMBL13660309 0.78 PDE4B (0.43) USP14PDE4BPDE4DOPRM1OPRL1
SCHEMBL13660453 0.76 SMN1; SMN2 (0.38) SMN1; SMN2PDE4BPDE7AGRM1
SCHEMBL13660351 0.74 SMN1; SMN2 (0.34) SMN1; SMN2PDE4BPDE7AGRM1
SCHEMBL3169334 0.72 PDE4B (0.33) SMN1; SMN2PDE4BPDE7A
SCHEMBL3169324 0.72 PDE4B (0.33) SMN1; SMN2PDE4BPDE7A
SCHEMBL13660314 0.69 PDE4B (0.34) DPP4USP14PDE4BPDE4D
SCHEMBL4755607 0.68 PDE4B (0.34) DPP4USP14PDE4BPDE4DOPRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009121036-A2 SUBSTITUTED ARYL PYRIMIDINONE DERIVATIVES NEUROGEN CORPORATION (US) 2009-10-01 WO disclosed