SCHEMBL13663151

SCHEMBL13663151

Cc1ccc(-c2nc(CBr)c(Br)s2)cc1

nearest known ligand 0.46

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.41
GAA P10253 3/20 0.41
RAB9A P51151 2/20 0.41
ALOX5 P09917 5/20 0.41
ALDH1A1 P00352 5/20 0.40
LMNA P02545 3/20 0.40
SMN1; SMN2 Q16637 3/20 0.40
TRPM8 Q7Z2W7 1/20 0.39
MAPT P10636 4/20 0.39
COMT P21964 1/20 0.38
APP P05067 2/20 0.36
NPC1 O15118 1/20 0.36
GLA P06280 1/20 0.36
TP53 P04637 1/20 0.36
KMT2A Q03164 2/20 0.36
HTT P42858 1/20 0.36
MEN1 O00255 1/20 0.36
SREBF2 Q12772 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13663143 0.85 PTGDR2 (0.43) KDM4EGAARAB9AALDH1A1LMNA
SCHEMBL1506655 0.82 PTGDR2 (0.42) KDM4EALDH1A1SMN1; SMN2MAPTKMT2A
SCHEMBL4051181 0.82 APP (0.50) KDM4EGAARAB9AALDH1A1SMN1; SMN2
SCHEMBL13654523 0.75 APP (0.44) RAB9ASMN1; SMN2APP
SCHEMBL13654522 0.74 PTGDR2 (0.36) APP
SCHEMBL13801070 0.73 ALOX5 (0.53) KDM4EGAARAB9AALOX5ALDH1A1
SCHEMBL13663150 0.72 TRPM8 (0.41) KDM4EGAARAB9AALDH1A1LMNA
SCHEMBL3370247 0.71 MAPT (0.51) KDM4EGAARAB9AALDH1A1SMN1; SMN2
SCHEMBL14417422 0.70 PTGDR2 (0.44) KDM4EALDH1A1SMN1; SMN2TRPM8MAPT
SCHEMBL1436257 0.70 HRH3 (0.46) GAAALOX5ALDH1A1SMN1; SMN2MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20090270447-A1 2-Aryl-and 2-Heteroarylthiazolyl Compounds, Methods for Their Preparation and Use Thereof WYETH (US) 2009-10-29 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090270447-A1 2-Aryl-and 2-Heteroarylthiazolyl Compounds, Methods for Their Preparation and Use Thereof CYP2U1, SEC22B, SEC63 KDM4E 3480/4885GAA 1533/4885RAB9A 1910/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.