SCHEMBL13664758

SCHEMBL13664758

COC(=O)c1ccc2[nH]c(=O)c(CN(CCc3ccccc3)C(=O)Nc3ccccc3)cc2c1

nearest known ligand 0.65

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
TSHR P16473 3/20 0.65
KDM4E B2RXH2 12/20 0.62
HSD17B10 Q99714 8/20 0.62
ALDH1A1 P00352 8/20 0.62
HPGD P15428 7/20 0.62
MAPT P10636 3/20 0.62
MEN1 O00255 3/20 0.62
KMT2A Q03164 3/20 0.62
CYP1A2 P05177 1/20 0.60
CYP3A4 P08684 1/20 0.60
CYP2D6 P10635 1/20 0.60
CYP2C9 P11712 1/20 0.60
CYP2C19 P33261 1/20 0.60
NPSR1 Q6W5P4 3/20 0.59
MAPK1 P28482 2/20 0.58
POLB P06746 1/20 0.55
GAA P10253 1/20 0.54
SMN1; SMN2 Q16637 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13665093 0.89 TSHR (0.61) TSHRKDM4EHSD17B10ALDH1A1HPGD
SCHEMBL13664756 0.85 TSHR (0.64) TSHRKDM4EHSD17B10ALDH1A1HPGD
SCHEMBL15270604 0.78 HDAC1 (0.72) KDM4EALDH1A1MAPTMEN1KMT2A
SCHEMBL18424429 0.74 KDM4E (0.78) TSHRKDM4EHSD17B10ALDH1A1HPGD
SCHEMBL13664838 0.72 KDM4E (0.70) KDM4EHSD17B10ALDH1A1HPGDMAPT
SCHEMBL13664590 0.71 KDM4E (0.69) KDM4EHSD17B10ALDH1A1HPGDMAPT
SCHEMBL13664841 0.71 KDM4E (0.68) KDM4EHSD17B10ALDH1A1HPGDMAPT
SCHEMBL13664845 0.70 KDM4E (0.66) TSHRKDM4EHSD17B10ALDH1A1HPGD
SCHEMBL4250505 0.69 ALDH1A1 (0.78) KDM4EHSD17B10ALDH1A1HPGDMAPT
SCHEMBL978722 0.68 F2 (0.62) KDM4EHPGDMEN1KMT2ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009128262-A1 QUINOLONE DERIVATIVE AND USE THEREOF 武田薬品工業株式会社 (JP) 2009-10-22 WO disclosed