SCHEMBL13670872

SCHEMBL13670872

O=C1CC[C@H](c2cccc(OC(F)(F)F)c2)N1c1ccccc1

nearest known ligand 0.47

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 4/20 0.47
HDAC6 Q9UBN7 4/20 0.47
HDAC8 Q9BY41 3/20 0.47
NOTUM Q6P988 1/20 0.46
CETP P11597 9/20 0.44
HDAC5 Q9UQL6 2/20 0.43
HCRTR1 O43613 3/20 0.43
HCRTR2 O43614 3/20 0.43
PIK3C3 Q8NEB9 2/20 0.41
DRD2 P14416 1/20 0.40
DRD3 P35462 1/20 0.40
KCNH2 Q12809 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13010992 0.90 MGLL (0.43) HDAC1HDAC6HDAC8CETPHDAC5
SCHEMBL27778845 0.90 HDAC1 (0.44) HDAC1HDAC6HDAC8NOTUMCETP
SCHEMBL13011721 0.87 CETP (0.41) HDAC1HDAC6HDAC8CETPHDAC5
SCHEMBL14155611 0.86 HDAC1 (0.55) HDAC1HDAC6HDAC8HDAC5HCRTR1
SCHEMBL2691178 0.83 TNKS (0.49) HDAC1HDAC6HDAC8HDAC5HCRTR1
SCHEMBL2693640 0.83 TNKS (0.49) HDAC1HDAC6HDAC8HDAC5HCRTR1
SCHEMBL2691174 0.83 TNKS (0.49) HDAC1HDAC6HDAC8HDAC5HCRTR1
SCHEMBL3739324 0.78 HDAC6 (0.54) HDAC1HDAC6HDAC8NOTUMHDAC5
SCHEMBL27778619 0.78 CETP (0.42) HDAC1HDAC6HDAC8CETPPIK3C3
SCHEMBL3586830 0.73 ALDH1A1 (0.47) DRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009131814-A2 1,5-DIPHENYL-PYRROLIDIN-2-ONE COMPOUNDS AS CB-1 LIGANDS ELI LILLY AND COMPANY (US) 2009-10-29 WO disclosed