SCHEMBL13675120

SCHEMBL13675120

CC(C)(C)OC(=O)N1C[C@@H](N)C[C@H]1C(=O)Nc1ccc(-n2ccncc2=O)cc1F

nearest known ligand 0.45

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.45
POLB P06746 1/20 0.45
CYP3A4 P08684 1/20 0.45
CYP2C19 P33261 1/20 0.45
F10 P00742 18/20 0.43
KCNH2 Q12809 1/20 0.39
ABL1 P00519 1/20 0.36
BCR P11274 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4496265 0.87 F10 (0.56) F10
SCHEMBL4490093 0.82 F10 (0.50) F10
SCHEMBL13674854 0.80 F10 (0.45) F10KCNH2
SCHEMBL13674873 0.80 F10 (0.41) F10KCNH2
SCHEMBL13674870 0.79 F10 (0.62) F10
SCHEMBL13675123 0.79 F10 (0.43) F10KCNH2
SCHEMBL13675102 0.78 F10 (0.46) F10KCNH2
SCHEMBL13675146 0.77 F10 (0.45) CYP1A2POLBCYP3A4CYP2C19F10
SCHEMBL4961883 0.77 F10 (0.70) F10
SCHEMBL3552468 0.73 F10 (0.41) POLBF10KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7601752-B2 Pyrrolidine derivatives HOFFMANN-LA ROCHE INC. (US) 2009-10-13 US disclosed