SCHEMBL13676258

SCHEMBL13676258

CC(=O)OC(COc1ccc(C)cc1)Cn1c(C(=O)OC(C)(C)C)cc2ccccc21

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
POLB P06746 4/20 0.44
MAPT P10636 2/20 0.44
NOD2 Q9HC29 3/20 0.44
NOD1 Q9Y239 3/20 0.44
KDM4E B2RXH2 3/20 0.44
KMT2A Q03164 3/20 0.43
THRB P10828 1/20 0.43
MEN1 O00255 2/20 0.40
NPSR1 Q6W5P4 2/20 0.40
LMNA P02545 1/20 0.40
CYP1A2 P05177 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2D6 P10635 1/20 0.40
CYP2C9 P11712 1/20 0.40
CYP2C19 P33261 1/20 0.40
RECQL P46063 1/20 0.40
NR1H2 P55055 1/20 0.39
GAA P10253 1/20 0.37
AR P10275 1/20 0.37
CRHBP P24387 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13676256 0.86 LMNA (0.56) POLBMAPTNOD2NOD1KDM4E
SCHEMBL3931693 0.86 PLA2G4A (0.52) POLBMAPTNOD2NOD1KMT2A
SCHEMBL13676280 0.79 MAPT (0.45) POLBMAPTKDM4EKMT2ATHRB
SCHEMBL13676257 0.78 PLA2G4A (0.54) MAPTNOD2NOD1KDM4EKMT2A
SCHEMBL13675811 0.77 LMNA (0.51) POLBMAPTKDM4EKMT2ATHRB
SCHEMBL13676285 0.73 AR (0.42) POLBMAPTKDM4EKMT2ATHRB
SCHEMBL28156129 0.73 KMT2A (0.46) POLBNOD2NOD1KDM4EKMT2A
SCHEMBL3929497 0.73 PLA2G4A (0.55) MAPTTHRBLMNACYP2D6NR1H2
SCHEMBL319362 0.70 CNR2 (0.52) POLBNOD2NOD1KDM4EKMT2A
SCHEMBL19410240 0.70 KMT2A (0.52) POLBNOD2NOD1KDM4EKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7608633-B2 Heteroaryl-substituted acetone derivatives as inhibitors of phospholipase A2 MERCKLE GMBH (DE) 2009-10-27 US disclosed