SCHEMBL13679677

SCHEMBL13679677

OC(O)c1ccc(/C=C/CBr)cc1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRIK1 P39086 2/20 0.33
GRIK2 Q13002 2/20 0.33
KDM4E B2RXH2 1/20 0.32
MAPK1 P28482 1/20 0.32
PTGS2 P35354 2/20 0.32
BCHE P06276 1/20 0.32
ACHE P22303 1/20 0.32
PAM P19021 1/20 0.31
NPC1 O15118 1/20 0.31
POLB P06746 1/20 0.31
RAB9A P51151 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
CYP3A4 P08684 2/20 0.31
MEN1 O00255 1/20 0.31
CYP2D6 P10635 1/20 0.31
MAPT P10636 1/20 0.31
CYP2C9 P11712 1/20 0.31
CYP2C19 P33261 1/20 0.31
KMT2A Q03164 1/20 0.31
PTGS1 P23219 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18821936 0.82 ALDH1A1 (0.41) PAMCYP3A4ALDH1A1RECQLCYP4F2
SCHEMBL13679671 0.81 ALDH1A1 (0.48) GRIK1GRIK2KDM4EMAPK1PTGS2
SCHEMBL3595590 0.79 KDM4E (0.48) GRIK1GRIK2KDM4EMAPK1PTGS2
SCHEMBL3595592 0.79 KDM4E (0.48) GRIK1GRIK2KDM4EMAPK1PTGS2
SCHEMBL9714628 0.76 ALDH1A1 (0.52) GRIK1GRIK2PTGS2PAMCYP3A4
SCHEMBL9714638 0.76 ALDH1A1 (0.52) GRIK1GRIK2PTGS2PAMCYP3A4
SCHEMBL9714631 0.76 ALDH1A1 (0.52) GRIK1GRIK2PTGS2PAMCYP3A4
SCHEMBL3466529 0.73 CYP2C19 (0.43) GRIK1GRIK2KDM4ERAB9ACYP3A4
SCHEMBL3466530 0.73 CYP2C19 (0.43) GRIK1GRIK2KDM4ERAB9ACYP3A4
SCHEMBL2451125 0.71 NFE2L2 (0.50) GRIK1GRIK2PTGS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0999835-B1 IMIDAZOLE DERIVATIVES AS MDR MODULATORS TAIJI BIOMEDICAL INC (US) 2009-09-09 EP disclosed
EP-2082740-A2 Use of imidazole derivatives as MDR modulators Taiji Biomedical, Inc. (US) 2009-07-29 EP disclosed