SCHEMBL13679682

SCHEMBL13679682

Cc1ccc(C(=O)C(=O)c2ccc(CBr)cc2)cc1

nearest known ligand 0.68

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CES2 O00748 5/20 0.68
CES1 P23141 5/20 0.68
GSK3B P49841 1/20 0.55
ALDH1A1 P00352 5/20 0.48
LMNA P02545 2/20 0.48
SRD5A2 P31213 1/20 0.47
SMN1; SMN2 Q16637 2/20 0.46
NPC1 O15118 4/20 0.46
RAB9A P51151 4/20 0.46
L3MBTL1 Q9Y468 1/20 0.46
KMT2A Q03164 3/20 0.43
PKM P14618 2/20 0.43
HTT P42858 2/20 0.43
ATM Q13315 2/20 0.43
NPSR1 Q6W5P4 2/20 0.43
MEN1 O00255 2/20 0.43
HPGD P15428 1/20 0.43
NLRP1 Q9C000 1/20 0.43
GAA P10253 1/20 0.43
NTSR1 P30989 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13679683 0.89 CES2 (0.83) CES2CES1ALDH1A1KMT2A
SCHEMBL7013140 0.88 ALDH1A1 (0.67) CES2CES1GSK3BALDH1A1LMNA
SCHEMBL121442 0.82
SCHEMBL167254 0.82 CES2 (1.00) CES2CES1GSK3BALDH1A1LMNA
SCHEMBL5734655 0.82 IDO1 (0.52) CES2CES1GSK3BALDH1A1TDP1
SCHEMBL12375837 0.81 CES2 (0.64) CES2CES1GSK3BALDH1A1LMNA
SCHEMBL1352549 0.81 CES2 (1.00) CES2CES1GSK3BALDH1A1LMNA
SCHEMBL28417303 0.81 CES2 (0.70) CES2CES1GSK3BALDH1A1LMNA
SCHEMBL20302436 0.79 IDO1 (0.50) CES2CES1GSK3BALDH1A1NPC1
SCHEMBL11030165 0.79 IDO1 (0.50) CES2CES1GSK3BALDH1A1TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0999835-B1 IMIDAZOLE DERIVATIVES AS MDR MODULATORS TAIJI BIOMEDICAL INC (US) 2009-09-09 EP disclosed
EP-2082740-A2 Use of imidazole derivatives as MDR modulators Taiji Biomedical, Inc. (US) 2009-07-29 EP disclosed