SCHEMBL7013140

SCHEMBL7013140

Cc1ccc(C(=O)c2ccc(CBr)cc2)cc1

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.67
LMNA P02545 2/20 0.67
SRD5A2 P31213 2/20 0.61
GSK3B P49841 1/20 0.55
CES2 O00748 2/20 0.52
CES1 P23141 2/20 0.52
RAB9A P51151 4/20 0.47
HTT P42858 3/20 0.47
SMN1; SMN2 Q16637 2/20 0.46
NPC1 O15118 3/20 0.46
L3MBTL1 Q9Y468 1/20 0.46
AKR1C3 P42330 1/20 0.44
PKM P14618 2/20 0.43
ATM Q13315 2/20 0.43
NPSR1 Q6W5P4 2/20 0.43
MEN1 O00255 2/20 0.43
KMT2A Q03164 2/20 0.43
HPGD P15428 1/20 0.43
NLRP1 Q9C000 1/20 0.43
GAA P10253 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9541276 0.89 CES2 (0.61) ALDH1A1LMNASRD5A2CES2CES1
SCHEMBL187134 0.89 CES2 (0.61) ALDH1A1LMNASRD5A2CES2CES1
SCHEMBL13679682 0.88 CES2 (0.68) ALDH1A1LMNASRD5A2GSK3BCES2
SCHEMBL10727688 0.83 SRD5A2 (0.85) ALDH1A1LMNASRD5A2GSK3BCES2
SCHEMBL11893040 0.83 SRD5A2 (0.85) ALDH1A1LMNASRD5A2GSK3BCES2
SCHEMBL5734655 0.82 IDO1 (0.52) ALDH1A1GSK3BCES2CES1TDP1
SCHEMBL52200 0.82 ALDH1A1 (1.00) ALDH1A1LMNASRD5A2CES2CES1
SCHEMBL822185 0.82 ALDH1A1 (1.00) ALDH1A1LMNASRD5A2CES2CES1
SCHEMBL121442 0.82
SCHEMBL118227 0.81 CES2 (0.77) ALDH1A1LMNASRD5A2GSK3BCES2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0733633-B1 Heterocyclic compounds, their production and use TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2003-05-28 EP disclosed
US-5753664-A ANTITUMOR AGENTS, PYRIMIDONES TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1998-05-19 US disclosed
EP-0733633-A1 Heterocyclic compounds, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1996-09-25 EP disclosed
US-5112851-A Agricultural Fungicides SANDOZ LTD. (CH) 1992-05-12 US disclosed
US-4939148-A Amine derivatives, processes for their production and their use SANDOZ, LTD. (CH) 1990-07-03 US disclosed