SCHEMBL13680725

SCHEMBL13680725

Cc1ccc(-c2ccc(=O)n(C)c2)o1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 2/20 0.51
ADORA1 P30542 2/20 0.51
ADORA3 P0DMS8 1/20 0.51
BRD4 O60885 7/20 0.41
DYRK1A Q13627 1/20 0.39
ADORA2B P29275 1/20 0.36
CREBBP Q92793 4/20 0.36
KDM4E B2RXH2 2/20 0.36
NPC1 O15118 2/20 0.36
ALDH1A1 P00352 2/20 0.36
LMNA P02545 2/20 0.36
HPGD P15428 2/20 0.36
RAB9A P51151 2/20 0.36
SMN1; SMN2 Q16637 2/20 0.36
GAA P10253 1/20 0.36
TSHR P16473 1/20 0.36
HSD17B10 Q99714 1/20 0.36
HSF1 Q00613 1/20 0.35
MAPT P10636 1/20 0.35
PKM P14618 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28463384 0.77 ADORA2A (0.55) ADORA2AADORA1ADORA3BRD4DYRK1A
SCHEMBL13680721 0.75 ADORA2A (0.43) ADORA2AADORA1ADORA3ADORA2BCREBBP
SCHEMBL22579156 0.74 ADORA2A (0.48) ADORA2AADORA1ADORA3BRD4ADORA2B
SCHEMBL23197679 0.73 TDP1 (0.56) KDM4ENPC1ALDH1A1LMNAHPGD
SCHEMBL29907698 0.73 ADORA2A (0.47) ADORA2AADORA1ADORA3ADORA2BKDM4E
SCHEMBL22552045 0.73 ADORA2A (0.47) ADORA2AADORA1ADORA3ADORA2BKDM4E
SCHEMBL29907757 0.72 ADORA2A (0.48) ADORA2AADORA1ADORA3BRD4DYRK1A
SCHEMBL13680601 0.72 TDP1 (0.39) KDM4ENPC1ALDH1A1LMNAHPGD
SCHEMBL16573986 0.71 BRD4 (0.50) BRD4DYRK1ACREBBP
SCHEMBL2319851 0.68 TDP1 (0.48) KDM4ENPC1ALDH1A1LMNAHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7582658-B2 Bicyclic compound ASAHI KASEI PHARMA CORPORATION (JP) 2009-09-01 US disclosed
US-7582658-B2 Bicyclic compound ASAHI KASEI PHARMA CORPORATION (JP) 2009-09-01 US disclosed